SCHEMBL20429656

SCHEMBL20429656

CCC1(C)CN(C(=O)CCO)CC1c1ccc(OC)c(OC2CN(c3ccc(C)cn3)C2)c1

nearest known ligand 0.54

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 17/20 0.54
PDE4A P27815 5/20 0.49
PDE4C Q08493 5/20 0.49
PDE4D Q08499 5/20 0.49
TACR3 P29371 2/20 0.42
PDE7A Q13946 1/20 0.41
CSF1R P07333 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18671554 1.00 PDE4B (0.54) PDE4BPDE4APDE4CPDE4DTACR3
SCHEMBL18872920 1.00 PDE4B (0.54) PDE4BPDE4APDE4CPDE4DTACR3
SCHEMBL19275958 0.92 PDE4B (0.64) PDE4BPDE4APDE4CPDE4DTACR3
SCHEMBL20429649 0.91 PDE4B (0.49) PDE4BPDE4APDE4CPDE4DTACR3
SCHEMBL18872625 0.91 PDE4B (0.49) PDE4BPDE4APDE4CPDE4DTACR3
SCHEMBL22152208 0.91 PDE4B (0.55) PDE4BPDE4APDE4CPDE4DTACR3
SCHEMBL18872918 0.89 PDE4B (0.68) PDE4BPDE4APDE4CPDE4DTACR3
SCHEMBL20429658 0.89 PDE4B (0.52) PDE4BPDE4APDE4CPDE4DPDE7A
SCHEMBL18873039 0.89 PDE4B (0.52) PDE4BPDE4APDE4CPDE4DPDE7A
SCHEMBL23956035 0.89 PDE4B (0.50) PDE4BPDE4APDE4CPDE4DTACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3189044-B1 CRYSTALLINE (2S)-3-[(3S,4S)-3-[(1R)-1-HYDROXYETHYL]-4-(4-METHOXY-3-{[1-(5-METHYLPYRIDIN-2-YL)AZETIDIN-3-YL]OXY}PHENYL) -3-METHYLPYRROLIDIN-1-YL]-3-OXOPROPANE-1,2-DIOL LILLY CO ELI (US) 2018-08-01 EP disclosed