SCHEMBL20458564

SCHEMBL20458564

CC(C)(C)OC(=O)N1CCN(c2nc(C3CC3)c(-c3cccnc3)cc2C#N)CC1C1CC1

nearest known ligand 0.44

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
RET P07949 1/20 0.44
IDH1 O75874 10/20 0.42
NR1H2 P55055 2/20 0.41
NR1H3 Q13133 2/20 0.41
GPR119 Q8TDV5 5/20 0.41
GBA1 P04062 1/20 0.40
KIT P10721 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14251107 1.00 RET (0.44) RETIDH1NR1H2NR1H3GPR119
SCHEMBL14251331 0.86 RET (0.43) RETIDH1NR1H2NR1H3GPR119
SCHEMBL14251333 0.86 RET (0.43) RETIDH1NR1H2NR1H3GPR119
SCHEMBL14251565 0.84 IDH1 (0.43) IDH1
SCHEMBL14315321 0.84 IDH1 (0.43) IDH1
SCHEMBL14251439 0.84 RET (0.42) RETIDH1NR1H2NR1H3GPR119
SCHEMBL14250774 0.84 RET (0.42) RETIDH1NR1H2NR1H3GPR119
SCHEMBL14250416 0.83 IDH1 (0.46) RETIDH1NR1H2NR1H3GPR119
SCHEMBL14250414 0.83 IDH1 (0.46) RETIDH1NR1H2NR1H3GPR119
SCHEMBL20458563 0.83 IDH1 (0.39) IDH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2721019-B1 THERAPEUTICALLY ACTIVE COMPOSITIONS AND THEIR METHODS OF USE AGIOS PHARMACEUTICALS INC (US) 2018-08-08 EP disclosed