SCHEMBL20458563

SCHEMBL20458563

CBN1CCN(c2nc(C3CC3)c(-c3cccnc3)cc2C#N)C[C@H]1C1CC1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 11/20 0.39
LRRK2 Q5S007 1/20 0.36
CFTR P13569 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
TSHR P16473 1/20 0.35
HSD17B10 Q99714 1/20 0.35
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
USP30 Q70CQ3 1/20 0.33
PIK3CD O00329 2/20 0.33
PIK3R1 P27986 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20458564 0.83 RET (0.44) IDH1
SCHEMBL14251107 0.83 RET (0.44) IDH1
SCHEMBL14251565 0.81 IDH1 (0.43) IDH1
SCHEMBL14315321 0.81 IDH1 (0.43) IDH1
SCHEMBL14318169 0.80 CHRNB2 (0.37) IDH1LRRK2CYP11B1CYP11B2USP30
SCHEMBL14250208 0.80 CHRNB2 (0.37) IDH1LRRK2CYP11B1CYP11B2USP30
SCHEMBL20458565 0.78 CYP1A2 (0.44) LRRK2CFTRALDH1A1CYP1A2CYP3A4
SCHEMBL15900550 0.73 IDH1 (0.50) IDH1PIK3CDPIK3R1
SCHEMBL14250708 0.73 IDH1 (0.50) IDH1PIK3CDPIK3R1
SCHEMBL14251607 0.73 IDH1 (0.51) IDH1PIK3CDPIK3R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2721019-B1 THERAPEUTICALLY ACTIVE COMPOSITIONS AND THEIR METHODS OF USE AGIOS PHARMACEUTICALS INC (US) 2018-08-08 EP disclosed