SCHEMBL20459338

SCHEMBL20459338

CC(C)(C)OC(C)(O)N1CCc2cc(N)ccc2C1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 1/20 0.50
ESR2 Q92731 7/20 0.42
HSD17B3 P37058 1/20 0.40
PDK2 Q15119 1/20 0.36
ESR1 P03372 6/20 0.35
DRD1 P21728 4/20 0.33
DRD5 P21918 3/20 0.33
DRD2 P14416 2/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
DRD3 P35462 1/20 0.33
MAPT P10636 1/20 0.33
TAAR1 Q96RJ0 1/20 0.33
BRD4 O60885 1/20 0.32
ATAD2 Q6PL18 1/20 0.32
KCNQ2 O43526 1/20 0.32
CA9 Q16790 1/20 0.32
HTR2A P28223 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13405609 0.82 NR1H2 (0.47) NR1H2ESR2HSD17B3PDK2ESR1
SCHEMBL17797585 0.75 NR1H2 (0.54) NR1H2HSD17B3PDK2DRD1DRD2
SCHEMBL61143 0.72 NR1H2 (0.90) NR1H2ESR2HSD17B3ESR1HDAC8
SCHEMBL29377835 0.72 NR1H2 (0.90) NR1H2ESR2HSD17B3ESR1HDAC8
SCHEMBL2510116 0.72 NR1H2 (0.53) NR1H2ESR2HSD17B3PDK2DRD1
SCHEMBL17797706 0.71 NR1H2 (0.44) NR1H2HSD17B3PDK2HDAC8HDAC6
SCHEMBL25856118 0.71 NR1H2 (0.49) NR1H2HSD17B3PDK2DRD1DRD2
SCHEMBL218317 0.70 MAOA (0.59) NR1H2HSD17B3DRD1DRD5DRD2
SCHEMBL30561544 0.70 MAOA (0.59) NR1H2HSD17B3DRD1DRD5DRD2
SCHEMBL6962549 0.70 HDAC6 (0.65) NR1H2ESR2HSD17B3ESR1HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2675793-B1 FAK INHIBITORS CANCER THERAPEUTICS CRC PTY LTD (AU) 2018-08-08 EP disclosed