SCHEMBL20459482

SCHEMBL20459482

CSc1cc(F)c(N)c(Br)c1

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.46
CA2 P00918 3/20 0.46
CA9 Q16790 3/20 0.46
ADRB2 P07550 10/20 0.38
MAPT P10636 2/20 0.36
GAA P10253 1/20 0.36
NPSR1 Q6W5P4 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
CA3 P07451 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3025702 0.77 HDAC1 (0.31) HDAC1HDAC6
SCHEMBL18398358 0.72 HTT (0.41) MAPT
SCHEMBL1394520 0.71 CA1 (0.50) CA1CA2CA9ADRB2MAPT
SCHEMBL1639935 0.70 CA1 (0.54) CA1CA2CA9ADRB2MAPT
SCHEMBL78688 0.70 CA1 (0.54) CA1CA2CA9ADRB2MAPT
SCHEMBL387740 0.70 KDM1A (0.37) MAPTGAA
SCHEMBL29504578 0.70 KDM1A (0.37) MAPTGAA
SCHEMBL15566427 0.70 IDO1 (0.36) MAPTGAANPSR1
SCHEMBL20079466 0.69 CES2 (0.36)
Hydrochloric Acid SCHEMBL7131081 0.69 CA1 (0.52) CA1CA2CA9ADRB2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3097083-B1 BENZIMIDAZOLE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF INFLAMMATORY DISORDERS GALAPAGOS NV (BE) 2018-08-08 EP disclosed