SCHEMBL20459581

SCHEMBL20459581

CCC(C)C(COC)c1ccc(F)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 2/20 0.37
SLC6A3 Q01959 2/20 0.37
AOC3 Q16853 1/20 0.37
SLC6A4 P31645 1/20 0.37
NOS3 P29474 1/20 0.36
NOS1 P29475 1/20 0.36
NOS2 P35228 1/20 0.36
LMNA P02545 3/20 0.35
ALDH1A1 P00352 2/20 0.35
IDO1 P14902 2/20 0.34
TDO2 P48775 2/20 0.34
MAPT P10636 2/20 0.34
ESR1 P03372 1/20 0.34
CYP1A2 P05177 1/20 0.34
PGR P06401 1/20 0.34
CHRM2 P08172 1/20 0.34
CYP3A4 P08684 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
AR P10275 1/20 0.34
CYP2D6 P10635 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2270719 0.85 AOC3 (0.43) SLC6A2SLC6A3AOC3SLC6A4LMNA
SCHEMBL15445213 0.83 AOC3 (0.43) SLC6A2SLC6A3AOC3SLC6A4LMNA
SCHEMBL17084072 0.83 AOC3 (0.43) SLC6A2SLC6A3AOC3SLC6A4LMNA
SCHEMBL25704721 0.83 AOC3 (0.43) SLC6A2SLC6A3AOC3SLC6A4LMNA
SCHEMBL12872171 0.83 ESR1 (0.45) SLC6A2SLC6A3AOC3LMNAALDH1A1
SCHEMBL19494020 0.81 TAAR1 (0.42) AOC3LMNAALDH1A1MAPTCHRM2
SCHEMBL17086661 0.75 AOC3 (0.42) SLC6A2SLC6A3AOC3SLC6A4LMNA
SCHEMBL17086659 0.75 AOC3 (0.42) SLC6A2SLC6A3AOC3SLC6A4LMNA
SCHEMBL16224877 0.75 AOC3 (0.42) SLC6A2SLC6A3AOC3SLC6A4LMNA
SCHEMBL15929826 0.74 AOC3 (0.42) SLC6A2SLC6A3AOC3SLC6A4NOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2900241-B1 NOVEL COMPOUNDS THAT ARE ERK INHIBITORS MERCK SHARP & DOHME (US) 2018-08-08 EP disclosed