SCHEMBL20459743

SCHEMBL20459743

O=NCc1ccc(F)cc1F

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.48
AGXT P21549 2/20 0.48
KDM4E B2RXH2 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
DAO P14920 1/20 0.41
HTR2A P28223 3/20 0.39
HTR2C P28335 3/20 0.39
MAOB P27338 1/20 0.39
CES2 O00748 1/20 0.39
CES1 P23141 1/20 0.39
RIPK1 Q13546 2/20 0.38
ALDH1A1 P00352 1/20 0.38
ATM Q13315 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
KCNH2 Q12809 1/20 0.36
GSK3B P49841 1/20 0.36
BACE1 P56817 1/20 0.36
MAPK8 P45983 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12028418 0.79 TP53 (0.42) IDO1HTR2AALDH1A1
SCHEMBL3483437 0.78 IDO1 (0.48) IDO1AGXTKDM4ESMN1; SMN2DAO
SCHEMBL14613820 0.78 IDO1 (0.48) IDO1AGXTKDM4ESMN1; SMN2DAO
SCHEMBL1647830 0.78 IDO1 (0.44) IDO1AGXTKDM4ESMN1; SMN2DAO
SCHEMBL15978572 0.75 IDO1 (0.50) IDO1AGXTKDM4ESMN1; SMN2DAO
SCHEMBL26699678 0.75
SCHEMBL518007 0.75 IDO1 (0.54) IDO1AGXTKDM4ESMN1; SMN2DAO
SCHEMBL469184 0.75 IDO1 (0.54) IDO1AGXTKDM4ESMN1; SMN2DAO
SCHEMBL7700904 0.74 IDO1 (0.58) IDO1AGXTKDM4ESMN1; SMN2DAO
SCHEMBL3298107 0.74 IDO1 (0.58) IDO1AGXTKDM4ESMN1; SMN2DAO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2721023-B1 METALLOENZYME INHIBITOR COMPOUNDS VIAMET PHARMACEUTICALS NC INC (US) 2018-08-08 EP disclosed