SCHEMBL20463333

SCHEMBL20463333

[O-][S+](c1ccc(OC(F)(F)F)cc1)N1CCC(c2nc3ccccc3[nH]2)CC1

nearest known ligand 0.60

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR2B P41595 5/20 0.60
TRPV1 Q8NER1 1/20 0.47
KMT2A Q03164 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.44
POLB P06746 1/20 0.43
MAPT P10636 1/20 0.43
ADRA1A P35348 2/20 0.43
KCNH2 Q12809 2/20 0.43
NPY5R Q15761 2/20 0.43
ALDH1A1 P00352 2/20 0.42
HTT P42858 1/20 0.42
PKM P14618 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20463309 0.86 HTR2B (0.58) HTR2BKMT2ASMN1; SMN2POLBMAPT
SCHEMBL20463474 0.86 HTR2B (0.48) HTR2BKMT2ASMN1; SMN2POLBMAPT
SCHEMBL20463432 0.85 KMT2A (0.62) HTR2BKMT2AALDH1A1PKM
SCHEMBL20463369 0.80 KMT2A (0.51) HTR2BKMT2AALDH1A1PKM
SCHEMBL20456432 0.80 KMT2A (0.74) HTR2BKMT2ASMN1; SMN2MAPTALDH1A1
SCHEMBL20463352 0.79 HTR2B (0.62) HTR2BTRPV1KMT2ASMN1; SMN2POLB
SCHEMBL1299510 0.75 HTR2B (1.00) HTR2BSMN1; SMN2
SCHEMBL13873294 0.75 SMN1; SMN2 (0.77) HTR2BTRPV1SMN1; SMN2POLBMAPT
SCHEMBL7950089 0.73 CARM1 (0.39) ALDH1A1
SCHEMBL7945321 0.73 CARM1 (0.39) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018144900-A1 SMALL MOLECULE ANTAGONISTS OF SUMO RELATED MODIFICATION OF CRMP2 AND USES THEREOF ARIZONA BOARD OF REGENTS ON BEHALF OF THE UNIVERSITY OF ARIZONA (US) 2018-08-09 WO disclosed