SCHEMBL20515841

SCHEMBL20515841

c1nc2c([nH]c3scnc32)s1

nearest known ligand 0.38

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DAO P14920 2/20 0.38
PI4KA P42356 1/20 0.34
PI4K2B Q8TCG2 1/20 0.34
PI4K2A Q9BTU6 1/20 0.34
PI4KB Q9UBF8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20631031 0.66
SCHEMBL20551383 0.63 CCR8 (0.34) DAO
SCHEMBL21578123 0.54 CSNK2A2 (0.33) PI4KAPI4K2BPI4K2API4KB
SCHEMBL21578110 0.54 PI4KA (0.31) PI4KAPI4K2BPI4K2API4KB
SCHEMBL12590225 0.50 MAPK1 (0.44)
SCHEMBL29360166 0.48 HSP90AA1 (0.39)
SCHEMBL29385656 0.48 HSP90AA1 (0.39)
SCHEMBL30358616 0.48 HSP90AA1 (0.39)
SCHEMBL29353635 0.48 HSP90AA1 (0.39)
SCHEMBL14380284 0.40 ALDH1A1 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10927214-B2 Method of making a pyrrolo bisthiazole homopolymer QATAR FOUNDATION FOR EDUCATION, SCIENCE AND COMMUNITY DEVELOPMENT (QA) 2021-02-23 US claimed
EP-3385298-B1 METHOD OF MAKING A PYRROLO BISTHIAZOLE HOMOPOLYMER QATAR FOUND EDUCATION SCIENCE & COMMUNITY DEV (QA) 2019-10-30 EP claimed
US-20190218337-A9 METHOD OF MAKING A PYRROLO BISTHIAZOLE HOMOPOLYMER QATAR FOUNDATION FOR EDUCATION, SCIENCE AND COMMUNITY DEVELOPMENT (QA) 2019-07-18 US claimed
EP-3385298-A1 METHOD OF MAKING A PYRROLO BISTHIAZOLE HOMOPOLYMER Qatar Foundation For Education Science And Community Development (QA) 2018-10-10 EP claimed
US-20180282473-A1 METHOD OF MAKING A PYRROLO BISTHIAZOLE HOMOPOLYMER QATAR FOUND EDUCATION SCIENCE & COMMUNITY DEV (QA) 2018-10-04 US claimed
EP-2630179-B1 CONJUGATED POLYMERS RAYNERGY TEK INC (TW) 2021-04-14 EP disclosed
US-10927214-B2 Method of making a pyrrolo bisthiazole homopolymer QATAR FOUNDATION FOR EDUCATION, SCIENCE AND COMMUNITY DEVELOPMENT (QA) 2021-02-23 US disclosed
US-10927214-B2 Method of making a pyrrolo bisthiazole homopolymer QATAR FOUNDATION FOR EDUCATION, SCIENCE AND COMMUNITY DEVELOPMENT (QA) 2021-02-23 US disclosed
EP-3385298-B1 METHOD OF MAKING A PYRROLO BISTHIAZOLE HOMOPOLYMER QATAR FOUND EDUCATION SCIENCE & COMMUNITY DEV (QA) 2019-10-30 EP disclosed
US-20190218337-A9 METHOD OF MAKING A PYRROLO BISTHIAZOLE HOMOPOLYMER QATAR FOUNDATION FOR EDUCATION, SCIENCE AND COMMUNITY DEVELOPMENT (QA) 2019-07-18 US disclosed
US-20190218337-A9 METHOD OF MAKING A PYRROLO BISTHIAZOLE HOMOPOLYMER QATAR FOUNDATION FOR EDUCATION, SCIENCE AND COMMUNITY DEVELOPMENT (QA) 2019-07-18 US disclosed
EP-3385298-A1 METHOD OF MAKING A PYRROLO BISTHIAZOLE HOMOPOLYMER Qatar Foundation For Education Science And Community Development (QA) 2018-10-10 EP disclosed
EP-3385298-A1 METHOD OF MAKING A PYRROLO BISTHIAZOLE HOMOPOLYMER Qatar Foundation For Education Science And Community Development (QA) 2018-10-10 EP disclosed
US-20180282473-A1 METHOD OF MAKING A PYRROLO BISTHIAZOLE HOMOPOLYMER QATAR FOUND EDUCATION SCIENCE & COMMUNITY DEV (QA) 2018-10-04 US disclosed
US-20180282473-A1 METHOD OF MAKING A PYRROLO BISTHIAZOLE HOMOPOLYMER QATAR FOUND EDUCATION SCIENCE & COMMUNITY DEV (QA) 2018-10-04 US disclosed