SCHEMBL20520529

SCHEMBL20520529

C#Cc1cnc2c(C)cc(OC(CC)(CC)C(N)=O)cc2c1

nearest known ligand 0.41

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.41
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22528909 0.88 PARP1 (0.40) PARP1
SCHEMBL21723834 0.86 PARP1 (0.39) PARP1
SCHEMBL29564411 0.86 PARP1 (0.39) PARP1
SCHEMBL23780875 0.82 PARP1 (0.38) PARP1
SCHEMBL20534741 0.82 PARP1 (0.38) PARP1
SCHEMBL23780868 0.81 PARP1 (0.40) PARP1
SCHEMBL23780882 0.79 PARP1 (0.37) PARP1
SCHEMBL20534739 0.78 PARP1 (0.38) PARP1
SCHEMBL18112844 0.78 PARP1 (0.41) PARP1
SCHEMBL21247562 0.78 PARP1 (0.34) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 45 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3978504-A1 CHIRAL 2,3-DIHYDROTHIAZOLO[3,2-A]PYRIMIDINE DERIVATIVES FOR COMBATING ANIMAL PESTS BASF SE (DE) 2022-04-06 EP claimed
US-20220046925-A1 METHOD OF CONTROLLING PESTS BY SEED TREATMENT APPLICATION OF A MESOIONIC COMPOUND OR MIXTURE THEREOF BASF SE (DE) 2022-02-17 US claimed
EP-3601298-B1 PROCESS FOR PREPARING CHIRAL 2,3-DIHYDROTHIAZOLO[3,2-A]PYRIMIDIN-4-IUM COMPOUNDS BASF SE (DE) 2021-12-01 EP claimed
US-20210355139-A1 Pyrimidinium Compounds and Their Mixtures for Combating Animal Pests BASF SE (DE) 2021-11-18 US claimed
WO-2020064492-A1 METHOD OF CONTROLLING PESTS BY SEED TREATMENT APPLICATION OF A MESOIONIC COMPOUND OR MIXTURE THEREOF BASF SE (DE) 2020-04-02 WO claimed
EP-3628156-A1 METHOD FOR CONTROLLING PESTS OF SUGARCANE, CITRUS, RAPESEED, AND POTATO PLANTS BASF SE (DE) 2020-04-01 EP claimed
EP-3601298-A1 PROCESS FOR PREPARING CHIRAL 2,3-DIHYDROTHIAZOLO[3,2-A]PYRIMIDIN-4-IUM COMPOUNDS BASF SE (DE) 2020-02-05 EP claimed
WO-2018177970-A1 PROCESS FOR PREPARING CHIRAL 2,3-DIHYDROTHIAZOLO[3,2-A]PYRIMIDIN-4-IUM COMPOUNDS BASF SE (DE) 2018-10-04 WO claimed
EP-3694852-B1 IMIDAZOLIDINE PYRIMIDINIUM COMPOUNDS FOR COMBATING ANIMAL PESTS BASF SE (DE) 2026-05-06 EP disclosed
US-20250255301-A1 PESTICIDAL MIXTURES COMPRISING A PYRAZOLE COMPOUND BASF SE (DE) 2025-08-14 US disclosed
EP-4486128-A1 COMPOSITIONS AND METHODS FOR TARGETED DELIVERY OF CHEMICALS AND BIOMOLECULES TO PLANTS AND FUNGI THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2025-01-08 EP disclosed
US-20240196908-A1 COMPOSITIONS AND METHODS FOR IMPROVING PLANT HEALTH AND CONTROLLING PLANT DISEASE AgBiome, Inc. (US) 2024-06-20 US disclosed
WO-2023168125-A1 COMPOSITIONS AND METHODS FOR TARGETED DELIVERY OF CHEMICALS AND BIOMOLECULES TO PLANTS AND FUNGI THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2023-09-07 WO disclosed
US-20230159562-A1 PYRIMIDINIUM COMPOUNDS AND THEIR MIXTURES FOR COMBATING ANIMAL PESTS BASF SE (DE) 2023-05-25 US disclosed
WO-2019175712-A1 NEW USES FOR CATECHOL MOLECULES AS INHIBITORS TO GLUTATHIONE S-TRANSFERASE METABOLIC PATHWAYS BASF CORPORATION (US) 2019-09-19 WO disclosed
WO-2019072906-A1 IMIDAZOLIDINE PYRIMIDINIUM COMPOUNDS FOR COMBATING ANIMAL PESTS BASF SE (DE) 2019-04-18 WO disclosed
EP-3453706-A1 PESTICIDAL IMIDAZOLE COMPOUNDS BASF SE (DE) 2019-03-13 EP disclosed
WO-2019042932-A1 METHOD OF CONTROLLING RICE PESTS IN RICE BASF SE (DE) 2019-03-07 WO disclosed
WO-2019043183-A1 METHOD OF CONTROLLING RICE PESTS IN RICE BASF SE (DE) 2019-03-07 WO disclosed
WO-2018177970-A1 PROCESS FOR PREPARING CHIRAL 2,3-DIHYDROTHIAZOLO[3,2-A]PYRIMIDIN-4-IUM COMPOUNDS BASF SE (DE) 2018-10-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230159562-A1 PYRIMIDINIUM COMPOUNDS AND THEIR MIXTURES FOR COMBATING ANIMAL PESTS THOP1, NIT2, DDT PARP1 2243/4885MAPT 1250/4885
US-20250255301-A1 PESTICIDAL MIXTURES COMPRISING A PYRAZOLE COMPOUND CYP51A1, CYP2S1, OSBP PARP1 4164/4885MAPT 3409/4885
US-20220046925-A1 METHOD OF CONTROLLING PESTS BY SEED TREATMENT APPLICATION OF A MESOIONIC COMPOUND OR MIXTURE THEREOF MANBA, CMA1, MTX1 PARP1 4858/4885MAPT 755/4885
US-20210355139-A1 Pyrimidinium Compounds and Their Mixtures for Combating Animal Pests THOP1, NIT2, DDT PARP1 2444/4885MAPT 1118/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.