SCHEMBL20523667

SCHEMBL20523667

CCCS(=O)(=O)Nc1cc(-c2cc(-c3ccc(N4CCNCC4)cc3)cnc2N)cc(Cl)c1OC

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NOD2 Q9HC29 16/20 1.00
ACVR1 Q04771 16/20 1.00
RIPK2 O43353 15/20 1.00
NOD1 Q9Y239 1/20 0.83
TGFBR1 P36897 3/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20523489 0.91 NOD2 (1.00) NOD2ACVR1RIPK2NOD1TGFBR1
SCHEMBL21630435 0.91 NOD2 (1.00) NOD2ACVR1RIPK2NOD1TGFBR1
SCHEMBL20523499 0.91 NOD2 (1.00) NOD2ACVR1RIPK2NOD1TGFBR1
SCHEMBL20523451 0.90 NOD2 (0.91) NOD2ACVR1RIPK2NOD1TGFBR1
SCHEMBL21630378 0.90 NOD2 (0.81) NOD2ACVR1RIPK2NOD1TGFBR1
SCHEMBL20523577 0.87 NOD2 (0.84) NOD2ACVR1RIPK2NOD1TGFBR1
SCHEMBL20523447 0.87 NOD2 (1.00) NOD2ACVR1RIPK2NOD1TGFBR1
SCHEMBL21630430 0.86 ACVR1 (1.00) NOD2ACVR1RIPK2NOD1TGFBR1
SCHEMBL20523618 0.84 NOD2 (0.84) NOD2ACVR1RIPK2NOD1
SCHEMBL21630444 0.84 NOD2 (1.00) NOD2ACVR1RIPK2NOD1TGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3600307-B1 COMPOSITIONS FOR USE IN METHODS OF INHIBITING PROTEIN KINASES UNIV HOUSTON SYSTEM (US) 2021-05-05 EP disclosed
EP-3600307-A1 COMPOSITIONS FOR USE IN METHODS OF INHIBITING PROTEIN KINASES University of Houston System (US) 2020-02-05 EP disclosed
WO-2018183633-A1 COMPOSITIONS FOR USE IN METHODS OF INHIBITING PROTEIN KINASES UNIVERSITY OF HOUSTON SYSTEM (US) 2018-10-04 WO disclosed