Cefotiam

Cefotiam

SCHEMBL20528733

CN(C)CCn1nnnc1SCC1=C(C(=O)O)N2C(=O)[C@@H](NC(=O)Cc3csc(N)n3)[C@H]2SC1.Cl.Cl.O

nearest known ligand 0.99

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

dacAdacBdacCftsImrcAmrcBmrdA

The experimentally established mechanism targets of Cefotiam. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.99
TDP1 Q9NUW8 8/20 0.97
LMNA P02545 3/20 0.97
HSD17B10 Q99714 2/20 0.97
NR1I2 O75469 3/20 0.57
PGR P06401 3/20 0.57
KDM4E B2RXH2 1/20 0.57
MEN1 O00255 1/20 0.57
KMT2A Q03164 1/20 0.57
POLB P06746 9/20 0.54
MAPT P10636 7/20 0.54
SMN1; SMN2 Q16637 1/20 0.51
SLC22A6 Q4U2R8 3/20 0.50
SLC22A8 Q8TCC7 3/20 0.50
SLC22A11 Q9NSA0 3/20 0.50
CTDSP1 Q9GZU7 2/20 0.50
PPARG P37231 2/20 0.50
ALDH1A1 P00352 3/20 0.49
SLC6A4 P31645 1/20 0.49
DAO P14920 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cefotiam SCHEMBL28028493 1.00 L3MBTL1 (0.99) L3MBTL1TDP1LMNAHSD17B10NR1I2
Cefotiam SCHEMBL27715723 1.00 L3MBTL1 (0.99) L3MBTL1TDP1LMNAHSD17B10NR1I2
Cefotiam SCHEMBL28264248 1.00 L3MBTL1 (0.99) L3MBTL1TDP1LMNAHSD17B10NR1I2
Cefotiam SCHEMBL28031009 1.00 L3MBTL1 (0.99) L3MBTL1TDP1LMNAHSD17B10NR1I2
Cefotiam SCHEMBL11065530 0.99 L3MBTL1 (1.00) L3MBTL1TDP1LMNAHSD17B10NR1I2
Cefotiam SCHEMBL193845 0.99 L3MBTL1 (1.00) L3MBTL1TDP1LMNAHSD17B10NR1I2
Cefotiam SCHEMBL65480 0.99 L3MBTL1 (1.00) L3MBTL1TDP1LMNAHSD17B10NR1I2
Cefotiam SCHEMBL28422039 0.99 TDP1 (0.99) L3MBTL1TDP1LMNAHSD17B10NR1I2
Cefotiam SCHEMBL10899868 0.99 L3MBTL1 (1.00) L3MBTL1TDP1LMNAHSD17B10NR1I2
Cefotiam SCHEMBL28181212 0.99 TDP1 (0.99) L3MBTL1TDP1LMNAHSD17B10NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3607084-B1 A METHOD FOR TESTING ANTIMICROBIAL SUSCEPTIBILITY UNIV WESTERN AUSTRALIA (AU) 2024-05-01 EP disclosed
US-20210292807-A1 METHOD FOR TESTING ANTIMICROBIAL SUSCEPTIBILITY THE UNIVERSITY OF WESTERN AUSTRALIA (AU) 2021-09-23 US disclosed
EP-3607084-A1 A METHOD FOR TESTING ANTIMICROBIAL SUSCEPTIBILITY The University Of Western Australia (AU) 2020-02-12 EP disclosed
WO-2018184073-A1 A METHOD FOR TESTING ANTIMICROBIAL SUSCEPTIBILITY THE UNIVERSITY OF WESTERN AUSTRALIA (AU) 2018-10-11 WO disclosed