SCHEMBL2053382

SCHEMBL2053382

Nc1ncnc2nc(-c3ccc([AsH2])cc3)cc(-c3cccc(Br)c3)c12

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADK P55263 11/20 0.73
KDM4E B2RXH2 2/20 0.59
HPGD P15428 2/20 0.59
PPARG P37231 2/20 0.59
NR2E3 Q9Y5X4 2/20 0.59
NCOR2 Q9Y618 2/20 0.59
POLB P06746 1/20 0.59
MCL1 Q07820 1/20 0.59
CYP1A2 P05177 1/20 0.59
CYP2C9 P11712 1/20 0.59
CYP2C19 P33261 1/20 0.59
PTK2B Q14289 1/20 0.59
KMT2A Q03164 2/20 0.58
MEN1 O00255 1/20 0.58
ALDH1A1 P00352 1/20 0.58
MAPT P10636 1/20 0.58
ALOX15 P16050 1/20 0.58
TSHR P16473 1/20 0.58
CASP1 P29466 1/20 0.58
BLM P54132 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8127996 0.91 ADK (0.78) ADKKDM4EHPGDPPARGNR2E3
SCHEMBL2039883 0.90 ADK (0.77) ADKKDM4EHPGDPPARGNR2E3
SCHEMBL8139237 0.90 ADK (0.76) ADKKDM4EHPGDPPARGNR2E3
SCHEMBL2035586 0.88 HPGD (0.77) ADKKDM4EHPGDPPARGNR2E3
SCHEMBL8136472 0.88 ADK (0.73) ADKKDM4EHPGDPPARGNR2E3
SCHEMBL2041886 0.88 ADK (0.73) ADKKDM4EHPGDPPARGNR2E3
SCHEMBL8128209 0.88 ADK (0.73) ADKKDM4EHPGDPPARGNR2E3
SCHEMBL8140762 0.87 PPARG (0.76) ADKKDM4EHPGDPPARGNR2E3
SCHEMBL2032548 0.87 ADK (0.72) ADKKDM4EHPGDPPARGNR2E3
SCHEMBL8153562 0.85 ADK (0.70) ADKKDM4EHPGDPPARGNR2E3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2513298-A2 BETA-CELL REPLICATION PROMOTING COMPOUNDS AND METHODS OF THEIR USE President and Fellows of Harvard College (US) 2012-10-24 EP disclosed
WO-2011075665-A2 BETA-CELL REPLICATION PROMOTING COMPOUNDS AND METHODS OF THEIR USE PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2011-06-23 WO disclosed