SCHEMBL20534818

SCHEMBL20534818

NC(=O)c1oc2cc(-c3ccc(-c4ccc(O)cc4)cc3)ccc2c1N

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.50
ALDH1A1 P00352 4/20 0.50
HSD17B10 Q99714 4/20 0.50
HPGD P15428 3/20 0.50
PTPN1 P18031 2/20 0.43
ESR1 P03372 3/20 0.41
ESR2 Q92731 3/20 0.41
CYP3A4 P08684 2/20 0.41
MAPK1 P28482 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
MPO P05164 1/20 0.41
CYP19A1 P11511 1/20 0.41
MAOA P21397 1/20 0.41
MAOB P27338 1/20 0.41
QPCT Q16769 1/20 0.41
IP6K2 Q9UHH9 1/20 0.41
CA12 O43570 1/20 0.40
CA9 Q16790 1/20 0.40
LCK P06239 1/20 0.40
MAPT P10636 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20535054 1.00 KDM4E (0.50) KDM4EALDH1A1HSD17B10HPGDPTPN1
SCHEMBL20535441 0.91 KDM4E (0.50) KDM4EALDH1A1HSD17B10HPGDESR1
SCHEMBL20535434 0.89 KDM4E (0.51) KDM4EALDH1A1HSD17B10HPGDSMN1; SMN2
SCHEMBL13699672 0.88 KDM4E (0.50) KDM4EALDH1A1HSD17B10HPGDSMN1; SMN2
SCHEMBL20535680 0.88 KDM4E (0.61) KDM4EALDH1A1HSD17B10HPGDPTPN1
SCHEMBL20534989 0.87 KDM4E (0.49) KDM4EALDH1A1HSD17B10HPGDPTPN1
SCHEMBL20535050 0.87 SMN1; SMN2 (0.49) KDM4EALDH1A1HSD17B10HPGDSMN1; SMN2
SCHEMBL20534963 0.83 KDM4E (0.52) KDM4EALDH1A1HSD17B10HPGDCYP3A4
SCHEMBL20535051 0.83 KDM4E (0.46) KDM4EALDH1A1HSD17B10HPGDCYP3A4
SCHEMBL20534970 0.83 ALDH1A1 (0.46) KDM4EALDH1A1HSD17B10HPGDCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018189683-A1 BENZOFURAN DERIVATIVES FOR USE AS AMPK ACTIVATORS UNIVERSITA' DI PISA (IT) 2018-10-18 WO claimed
WO-2018189683-A1 BENZOFURAN DERIVATIVES FOR USE AS AMPK ACTIVATORS UNIVERSITA' DI PISA (IT) 2018-10-18 WO disclosed