SCHEMBL2053816

SCHEMBL2053816

O=C(O)c1cccc(CCl)c1[N+](=O)[O-]

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.49
TSHR P16473 4/20 0.49
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
MAPT P10636 2/20 0.40
HMGB1 P09429 1/20 0.40
PLA2G1B P04054 1/20 0.40
ATG4B Q9Y4P1 1/20 0.40
FOLH1 Q04609 1/20 0.40
CDK2 P24941 1/20 0.39
ALOX15 P16050 1/20 0.39
HPGD P15428 2/20 0.39
TP53 P04637 1/20 0.39
CYP1A2 P05177 2/20 0.38
CYP2C19 P33261 2/20 0.38
CYP2D6 P10635 1/20 0.38
POLB P06746 1/20 0.38
HSP90AA1 P07900 1/20 0.38
RAB9A P51151 1/20 0.38
CLCN2 P51788 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27535973 0.98 ALDH1A1 (0.47) ALDH1A1TSHRMEN1KMT2AMAPT
SCHEMBL27900413 0.87 TSHR (0.45) ALDH1A1TSHRMEN1KMT2AMAPT
SCHEMBL8708820 0.84 TSHR (0.49) ALDH1A1TSHRMEN1KMT2AMAPT
SCHEMBL8708824 0.84 TSHR (0.49) ALDH1A1TSHRMEN1KMT2AMAPT
SCHEMBL1523175 0.84 TSHR (0.53) ALDH1A1TSHRMEN1KMT2AMAPT
SCHEMBL25231628 0.83 HMGB1 (0.47) ALDH1A1TSHRMEN1KMT2AMAPT
SCHEMBL4369127 0.83 TSHR (0.47) ALDH1A1TSHRMEN1KMT2AMAPT
SCHEMBL25274950 0.83 TSHR (0.47) ALDH1A1TSHRMEN1KMT2AMAPT
SCHEMBL1497989 0.81 TSHR (0.60) ALDH1A1TSHRMEN1KMT2AMAPT
SCHEMBL28638919 0.81 TSHR (0.43) ALDH1A1TSHRMEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2326650-A2 DIHYDROPYRIDOPHTHALAZINONE INHIBITORS OF POLY(ADP-RIBOSE)POLYMERASE (PARP) BioMarin Pharmaceutical Inc. (US) 2011-06-01 EP disclosed
WO-2010017055-A2 DIHYDROPYRIDOPHTHALAZINONE INHIBITORS OF POLY(ADP-RIBOSE)POLYMERASE (PARP) LEAD THERAPEUTICS, INC. (US) 2010-02-11 WO disclosed