SCHEMBL20544375

SCHEMBL20544375

CCc1cc(=O)[nH]nc1Cc1ccc(F)c(C(=O)N2CCCNCC2)c1

nearest known ligand 0.70

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 20/20 0.70
PARP3 Q9Y6F1 1/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL3913847 0.95 PARP1 (0.64) PARP1PARP3
SCHEMBL20544232 0.86 PARP1 (0.74) PARP1PARP3
SCHEMBL20544273 0.85 PARP1 (0.73) PARP1PARP3
SCHEMBL20544379 0.85 PARP1 (0.72) PARP1PARP3
SCHEMBL20544383 0.84 PARP1 (0.77) PARP1PARP3
SCHEMBL20544688 0.84 PARP1 (0.68) PARP1PARP3
SCHEMBL4555783 0.82 PARP1 (1.00) PARP1PARP3
Trifluoroacetic Acid SCHEMBL3912153 0.82 PARP1 (0.68) PARP1PARP3
SCHEMBL864319 0.81 PARP1 (1.00) PARP1PARP3
SCHEMBL29434944 0.81 PARP1 (1.00) PARP1PARP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029551-B1 PYRIDINONE AND PYRIDAZINONE DERIVATIVES AS INHIBITORS OF POLY(ADP-RIBOSE)POLYMERASE (PARP) MSD ITALIA SRL (IT) 2018-10-31 EP claimed