SCHEMBL20544381

SCHEMBL20544381

COc1ccc(Cc2n[nH]c(=O)c(C)c2C)cc1C(=O)N1CCn2c(nnc2C(F)(F)F)C1

nearest known ligand 0.64

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 20/20 0.64
PARP2 Q9UGN5 1/20 0.57
PARP3 Q9Y6F1 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL3981579 0.98 PARP1 (0.61) PARP1PARP2PARP3
SCHEMBL20544501 0.92 PARP1 (0.61) PARP1PARP2PARP3
Trifluoroacetic Acid SCHEMBL4246186 0.90 PARP1 (0.59) PARP1PARP2PARP3
SCHEMBL4252874 0.90 PARP1 (0.78) PARP1
SCHEMBL20544235 0.88 PARP1 (0.64) PARP1PARP2PARP3
Trifluoroacetic Acid SCHEMBL4244887 0.85 PARP1 (0.61) PARP1PARP2PARP3
SCHEMBL20544497 0.84 PARP1 (0.79) PARP1PARP2PARP3
SCHEMBL3983235 0.83 PARP1 (0.69) PARP1
Trifluoroacetic Acid SCHEMBL4244891 0.82 PARP1 (0.76) PARP1PARP2PARP3
SCHEMBL3981582 0.82 PARP1 (0.48) PARP1PARP2PARP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029551-B1 PYRIDINONE AND PYRIDAZINONE DERIVATIVES AS INHIBITORS OF POLY(ADP-RIBOSE)POLYMERASE (PARP) MSD ITALIA SRL (IT) 2018-10-31 EP claimed