SCHEMBL3983235

SCHEMBL3983235

Cc1c(Cc2ccc(F)c(C(=O)N3CCn4c(nnc4C(F)(F)C(F)(F)F)C3)c2)n[nH]c(=O)c1C

nearest known ligand 0.69

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 20/20 0.69
KCNH2 Q12809 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL4241086 0.98 PARP1 (0.66) PARP1KCNH2
SCHEMBL4252874 0.94 PARP1 (0.78) PARP1
SCHEMBL20544662 0.89 PARP1 (0.68) PARP1
SCHEMBL19005624 0.88 PARP1 (0.88) PARP1KCNH2
Trifluoroacetic Acid SCHEMBL4247765 0.88 PARP1 (0.65) PARP1
Trifluoroacetic Acid SCHEMBL4248736 0.88 PARP1 (0.67) PARP1
SCHEMBL3985679 0.87 PARP1 (0.71) PARP1
SCHEMBL19005726 0.87 PARP1 (0.75) PARP1KCNH2
Trifluoroacetic Acid SCHEMBL3922864 0.86 PARP1 (0.61) PARP1
SCHEMBL20544671 0.86 PARP1 (0.63) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029551-B1 PYRIDINONE AND PYRIDAZINONE DERIVATIVES AS INHIBITORS OF POLY(ADP-RIBOSE)POLYMERASE (PARP) MSD ITALIA SRL (IT) 2018-10-31 EP claimed
EP-2029551-A2 PYRIDINONE AND PYRIDAZINONE DERIVATIVES AS INHIBITORS OF POLY(ADP-RIBOSE)POLYMERASE (PARP) ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI S.P.A. (IT) 2009-03-04 EP disclosed
WO-2007138351-A2 PYRIDINONE AND PYRIDAZINONE DERIVATIVES AS INHIBITORS OF POLY(ADP-RIBOSE)POLYMERASE (PARP) ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2007-12-06 WO disclosed