SCHEMBL20547726

SCHEMBL20547726

CC1(Nc2ncnc3cnccc23)COC1

nearest known ligand 0.62

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
LATS1 O95835 17/20 0.62
LATS2 Q9NRM7 8/20 0.62
EGFR P00533 2/20 0.46
MKNK1 Q9BUB5 1/20 0.42
MKNK2 Q9HBH9 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29707469 0.87 LATS1 (0.61) LATS1LATS2EGFR
SCHEMBL20547912 0.84 LATS1 (0.61) LATS1LATS2EGFR
SCHEMBL20547760 0.76 LATS1 (1.00) LATS1LATS2
SCHEMBL29650587 0.73 LATS1 (0.56) LATS1LATS2EGFR
SCHEMBL17142299 0.72 CYP1A2 (0.45) EGFR
SCHEMBL3322882 0.71 EGFR (0.56) LATS1LATS2EGFRMKNK1MKNK2
SCHEMBL22302812 0.70 LATS1 (0.56) LATS1LATS2EGFR
SCHEMBL31375184 0.70 EGFR (0.53) LATS1EGFRMKNK1MKNK2
SCHEMBL31375768 0.68 EGFR (0.65) LATS1EGFR
SCHEMBL29650589 0.68 EGFR (0.61) LATS1LATS2EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3615537-A2 6-6 FUSED BICYCLIC HETEROARYL COMPOUNDS AND THEIR USE AS LATS INHIBITORS Novartis AG (CH) 2020-03-04 EP disclosed
WO-2018198077-A2 6-6 FUSED BICYCLIC HETEROARYL COMPOUNDS AND THEIR USE AS LATS INHIBITORS NOVARTIS AG (CH) 2018-11-01 WO disclosed