Odapipam

Odapipam

SCHEMBL2056522

CN1CCc2cc(Cl)c(O)cc2[C@@H](c2cccc3c2OCC3)C1

nearest known ligand 0.66

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 12/20 0.66
DRD5 P21918 5/20 0.62
DRD2 P14416 3/20 0.62
CYP1A2 P05177 2/20 0.62
CYP2D6 P10635 2/20 0.62
TSHR P16473 2/20 0.62
HSD17B10 Q99714 2/20 0.62
CYP3A4 P08684 1/20 0.62
NFKB1 P19838 1/20 0.62
THPO P40225 1/20 0.62
MEN1 O00255 1/20 0.62
ALOX15 P16050 1/20 0.62
KMT2A Q03164 1/20 0.62
SIGMAR1 Q99720 1/20 0.62
LMNA P02545 1/20 0.61
ADRB2 P07550 1/20 0.61
GPR183 P32249 1/20 0.61
APLNR P35414 1/20 0.61
GLP1R P43220 1/20 0.61
CX3CR1 P49238 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Odapipam SCHEMBL7207803 1.00 DRD1 (0.66) DRD1DRD5DRD2CYP1A2CYP2D6
Odapipam SCHEMBL1230030 0.95 DRD1 (0.60) DRD1DRD5DRD2CYP1A2CYP2D6
SCHEMBL10695137 0.94 DRD1 (0.64) DRD1DRD5DRD2CYP1A2CYP2D6
SCHEMBL9404411 0.87 DRD1 (0.52) DRD1DRD5DRD2CYP1A2CYP2D6
SCHEMBL8911525 0.86 DRD1 (0.58) DRD1DRD5DRD2CYP1A2CYP2D6
SCHEMBL8911123 0.85 DRD1 (0.55) DRD1DRD5DRD2CYP1A2CYP2D6
SCHEMBL31257120 0.84 DRD1 (0.45) DRD1DRD5DRD2CYP1A2CYP2D6
SCHEMBL8911502 0.84 DRD1 (0.56) DRD1DRD5DRD2CYP1A2CYP2D6
SCHEMBL8911122 0.84 DRD1 (0.56) DRD1DRD5DRD2CYP1A2CYP2D6
Berupipam SCHEMBL7797350 0.84 DRD1 (0.56) DRD1DRD5DRD2CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 78 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024136579-A1 COMPOSITION FOR PREVENTING, AMELIORATING, OR TREATING COGNITIVE DYSFUNCTION, CONTAINING DOPAMINE PRODUCTION INHIBITOR OR DOPAMINE RECEPTOR ANTAGONIST 서울대학교산학협력단 2024-06-27 WO claimed
EP-1931320-B1 MICROPARTICLES WITH MODIFIED RELEASE OF AT LEAST ONE ACTIVE PRINCIPLE AND ORAL DOSAGE FORM COMPRISING THE SAME FLAMEL IRELAND LTD (IE) 2022-06-15 EP claimed
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US claimed
US-20100226943-A1 SURFACE TOPOGRAPHIES FOR NON-TOXIC BIOADHESION CONTROL UNIVERSITY OF FLORIDA (US) 2010-09-09 US claimed
US-20090220611-A1 Microparticles With Modified Release of At Least One Active Principle and Oral Pharmaceutical Form Comprising Same FLAMEL TECHNOLOGIES, S.A. (FR) 2009-09-03 US claimed
CN-101330905-A Freeze-drying process and products obtained thereby SCIDOSE LLC (US) 2008-12-24 CN claimed
EP-1954244-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY Scidose, Llc (US) 2008-08-13 EP claimed
EP-1931320-A2 MICROPARTICLES WITH MODIFIED RELEASE OF AT LEAST ONE ACTIVE PRINCIPLE AND ORAL GALENIC FORM COMPRISING SAME Flamel Technologies (FR) 2008-06-18 EP claimed
WO-2007061529-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY SCIDOSE LLC. (US) 2007-05-31 WO claimed
US-20070116729-A1 Lyophilization process and products obtained thereby SCIDOSE LLC 2007-05-24 US claimed
WO-2007036671-A2 MICROPARTICLES WITH MODIFIED RELEASE OF AT LEAST ONE ACTIVE PRINCIPLE AND ORAL GALENIC FORM COMPRISING SAME FLAMEL TECHNOLOGIES (FR) 2007-04-05 WO claimed
US-20250340671-A1 METHODS AND PHARMACEUTICAL COMPOSITIONS FOR REDUCING THE NEUROMODULATORY EFFECT OF COCAINE UNIVERSITY OF CINCINNATI (US) 2025-11-06 US disclosed
WO-2024136579-A1 COMPOSITION FOR PREVENTING, AMELIORATING, OR TREATING COGNITIVE DYSFUNCTION, CONTAINING DOPAMINE PRODUCTION INHIBITOR OR DOPAMINE RECEPTOR ANTAGONIST 서울대학교산학협력단 2024-06-27 WO disclosed
US-20220290159-A1 miRNAS FOR REDUCING VENTRICLE ENLARGEMENT St. Jude Children's Research Hpspital, Inc. (US) 2022-09-15 US disclosed
US-11389453-B2 Compositions and methods for treating chemosensory dysfunction CYRANO THERAPEUTICS, INC. (US) 2022-07-19 US disclosed
EP-1411901-A1 GASTRIC RETENTION CONTROLLED DRUG DELIVERY SYSTEM Sun Pharmaceuticals Industries Ltd. (IN) 2004-04-28 EP disclosed
WO-2003011255-A1 GASTRIC RETENTION CONTROLLED DRUG DELIVERY SYSTEM SUN PHARMACEUTICAL INDUSTRIES LIMITED (IN) 2003-02-13 WO disclosed
US-5760216-A REACTING DRUG SAMPLE WITH SYNTHETIC METALLOPORPHYRIN, OXIDIZING AGENT, SOLVENT TO FORM OXIDATION PRODUCT ABBOTT LABORATORIES (US) 1998-06-02 US disclosed
EP-0781261-A2 USE OF SYNTHETIC METALLOPORPHYRINS FOR PREPARATION AND PREDICTION OF DRUG METABOLITES Abbott Laboratories (US) 1997-07-02 EP disclosed
WO-1996008455-A2 USE OF SYNTHETIC METALLOPORPHYRINS FOR PREPARATION AND PREDICTION OF DRUG METABOLITES ABBOTT LABORATORIES (US) 1996-03-21 WO disclosed