SCHEMBL20570524

SCHEMBL20570524

COC(=O)c1cc(OC2CCN(C(=O)OC(C)(C)C)CC2)ccc1C(F)(F)F

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 7/20 0.54
EPHX2 P34913 1/20 0.52
ALDH1A1 P00352 1/20 0.47
HRH3 Q9Y5N1 1/20 0.47
NEK2 P51955 1/20 0.46
PDE4A P27815 1/20 0.45
PDE4B Q07343 1/20 0.45
PDE4C Q08493 1/20 0.45
PDE4D Q08499 1/20 0.45
CHEK2 O96017 1/20 0.44
STS P08842 1/20 0.44
EED O75530 1/20 0.44
RBBP4 Q09028 1/20 0.44
SUZ12 Q15022 1/20 0.44
EZH2 Q15910 1/20 0.44
AEBP2 Q6ZN18 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25206434 0.88 GPR119 (0.56) GPR119ALDH1A1HRH3PDE4APDE4B
SCHEMBL30612802 0.88 GPR119 (0.56) GPR119ALDH1A1HRH3PDE4APDE4B
SCHEMBL20570944 0.88 GPR119 (0.52) GPR119EPHX2ALDH1A1HRH3NEK2
SCHEMBL20570726 0.87 EPHX2 (0.42) GPR119EPHX2HRH3
SCHEMBL30344060 0.86 GPR119 (0.54) GPR119ALDH1A1HRH3PDE4APDE4B
SCHEMBL25155201 0.86 GPR119 (0.54) GPR119ALDH1A1HRH3PDE4APDE4B
SCHEMBL22265776 0.85 GPR119 (0.66) GPR119EPHX2ALDH1A1HRH3NEK2
SCHEMBL7356060 0.84 GPR119 (0.54) GPR119ALDH1A1HRH3PDE4APDE4B
SCHEMBL8088637 0.84 GPR119 (0.57) GPR119EPHX2ALDH1A1HRH3NEK2
SCHEMBL31071590 0.84 GPR119 (0.57) GPR119EPHX2HRH3NEK2CHEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3634404-B1 PYRAZOLE MAGL INHIBITORS H LUNDBECK AS (DK) 2024-11-20 EP disclosed
CN-110678177-B Pyrazole MAGL inhibitors H.隆德贝克有限公司 2023-06-13 CN disclosed
US-11149037-B2 Pyrazole MAGL inhibitors H. LUNDBECK A/S (DK) 2021-10-19 US disclosed
US-11149037-B2 Pyrazole MAGL inhibitors H. LUNDBECK A/S (DK) 2021-10-19 US disclosed
EP-3634404-A1 PYRAZOLE MAGL INHIBITORS Lundbeck La Jolla Research Center, Inc. (US) 2020-04-15 EP disclosed
US-20200087304-A1 PYRAZOLE MAGL INHIBITORS H. LUNDBECK A/S (DK) 2020-03-19 US disclosed
US-20200087304-A1 PYRAZOLE MAGL INHIBITORS H. LUNDBECK A/S (DK) 2020-03-19 US disclosed
CN-110678177-A Pyrazole MAGL inhibitors 隆德贝克拉荷亚研究中心有限公司 2020-01-10 CN disclosed
WO-2018217809-A1 PYRAZOLE MAGL INHIBITORS ABIDE THERAPEUTICS, INC. (US) 2018-11-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11149037-B2 Pyrazole MAGL inhibitors MAGI3, MAG, PYM1 GPR119 2756/4885EPHX2 2642/4885ALDH1A1 4019/4885
US-20200087304-A1 PYRAZOLE MAGL INHIBITORS MAGI3, MAG, PYM1 GPR119 2756/4885EPHX2 2642/4885ALDH1A1 4019/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.