SCHEMBL20588993

SCHEMBL20588993

O=C(NCc1ccccn1)Nc1cc(F)c(Oc2ccnc3[nH]cc(Br)c23)c(F)c1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TBK1 Q9UHD2 1/20 0.51
NPC1 O15118 5/20 0.49
KMT2A Q03164 4/20 0.49
MEN1 O00255 1/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
ALOX15 P16050 1/20 0.48
RAB9A P51151 5/20 0.47
MAPT P10636 2/20 0.45
GLA P06280 1/20 0.45
HTT P42858 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.44
TSHR P16473 1/20 0.44
HPGD P15428 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20588094 0.90 TBK1 (0.51) TBK1
SCHEMBL20589077 0.89 NPC1 (0.56) TBK1NPC1KMT2AMEN1SMN1; SMN2
SCHEMBL20588499 0.88 MAP4K1 (0.52) TBK1NPC1KMT2AMEN1SMN1; SMN2
SCHEMBL20588497 0.88 TBK1 (0.51) TBK1
SCHEMBL20588539 0.86 TBK1 (0.51) TBK1HTT
SCHEMBL20588016 0.86 TBK1 (0.49) TBK1
SCHEMBL20588160 0.84 TBK1 (0.50) TBK1
SCHEMBL20588124 0.84 TBK1 (0.53) TBK1
SCHEMBL20588709 0.84 KMT2A (0.51) NPC1KMT2AMEN1SMN1; SMN2ALOX15
SCHEMBL20589113 0.83 TBK1 (0.51) TBK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3638669-A1 SUBSTITUTED PYRROLOPYRIDINE-DERIVATIVES Bayer Pharma Aktiengesellschaft (DE) 2020-04-22 EP claimed
WO-2018228920-A1 SUBSTITUTED PYRROLOPYRIDINE-DERIVATIVES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-12-20 WO claimed
EP-3638669-A1 SUBSTITUTED PYRROLOPYRIDINE-DERIVATIVES Bayer Pharma Aktiengesellschaft (DE) 2020-04-22 EP disclosed
WO-2018228920-A1 SUBSTITUTED PYRROLOPYRIDINE-DERIVATIVES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-12-20 WO disclosed