SCHEMBL20596995

SCHEMBL20596995

CC(C)c1ccc2c(c1)-c1sc(C(N)=O)cc1CO2

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.55
GAA P10253 7/20 0.55
KDM4E B2RXH2 6/20 0.55
L3MBTL1 Q9Y468 3/20 0.55
NOTUM Q6P988 8/20 0.53
MAPT P10636 5/20 0.52
PIK3CA P42336 4/20 0.51
HPGD P15428 5/20 0.50
HSD17B10 Q99714 4/20 0.50
MAPK1 P28482 3/20 0.50
GLA P06280 3/20 0.49
CASP1 P29466 2/20 0.49
CASP7 P55210 2/20 0.49
TSHR P16473 1/20 0.49
ATM Q13315 1/20 0.49
HTT P42858 3/20 0.45
TP53 P04637 3/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
SMN1; SMN2 Q16637 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20597270 0.89 NOTUM (0.67) ALDH1A1GAAKDM4EL3MBTL1NOTUM
SCHEMBL28825316 0.82 NOTUM (0.57) ALDH1A1GAAKDM4EL3MBTL1NOTUM
SCHEMBL20597377 0.81 NOTUM (0.79) ALDH1A1GAAKDM4EL3MBTL1NOTUM
SCHEMBL988495 0.81 NOTUM (0.56) ALDH1A1GAAKDM4EL3MBTL1NOTUM
SCHEMBL20597428 0.81 NOTUM (0.79) ALDH1A1GAAKDM4EL3MBTL1NOTUM
SCHEMBL20597096 0.79 NOTUM (0.78) ALDH1A1GAAKDM4EL3MBTL1NOTUM
SCHEMBL20597503 0.76 NOTUM (0.63) ALDH1A1GAAKDM4EL3MBTL1NOTUM
SCHEMBL20597360 0.73 NOTUM (0.63) ALDH1A1GAAKDM4EL3MBTL1NOTUM
SCHEMBL20597320 0.73 MAPT (0.56) ALDH1A1GAAKDM4EL3MBTL1NOTUM
SCHEMBL989468 0.72 NOTUM (0.72) ALDH1A1GAAKDM4EL3MBTL1NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2714675-B1 4H-THIENO[3,2-C]CHROMENE-BASED INHIBITORS OF NOTUM PECTINACETYLESTERASE AND METHODS OF THEIR USE LEXICON PHARMACEUTICALS INC (US) 2019-01-02 EP disclosed