SCHEMBL20615744

SCHEMBL20615744

Cc1ncccc1OC(=O)N1CCC([C@@H](C)NC(=O)c2ccc(Cl)cc2)CC1

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 6/20 0.55
ALDH1A1 P00352 2/20 0.46
CHRNA1 P02708 1/20 0.45
CYP2C8 P10632 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
NAMPT P43490 2/20 0.45
GPR119 Q8TDV5 1/20 0.44
SMYD3 Q9H7B4 8/20 0.44
KDM4E B2RXH2 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CCR1 P32246 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20600971 0.91 ALDH1A1 (0.46) IDO1ALDH1A1NAMPTGPR119SMYD3
SCHEMBL20601136 0.89 IDO1 (0.49) IDO1ALDH1A1CYP2C9GPR119KDM4E
SCHEMBL20600950 0.89 IDO1 (0.49) IDO1ALDH1A1CYP2C9GPR119KDM4E
SCHEMBL20616363 0.89 IDO1 (0.53) IDO1ALDH1A1CHRNA1CYP2C8CYP2C9
SCHEMBL20600914 0.87 CCR1 (0.42) IDO1ALDH1A1CYP2C9CYP2C19GPR119
SCHEMBL20600913 0.87 CCR1 (0.42) IDO1ALDH1A1CYP2C9CYP2C19GPR119
SCHEMBL20600935 0.83 IDO1 (0.48) IDO1ALDH1A1CHRNA1CYP2C8CYP2C9
SCHEMBL20600934 0.83 IDO1 (0.48) IDO1ALDH1A1CHRNA1CYP2C8CYP2C9
SCHEMBL20615754 0.82 KDM4E (0.50) ALDH1A1NAMPTKDM4ESMN1; SMN2
SCHEMBL20601177 0.80 ALDH1A1 (0.45) IDO1ALDH1A1NAMPTSMYD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019003141-A1 MODULATORS OF INDOLEAMINE 2,3-DIOXYGENASE GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2019-01-03 WO disclosed