SCHEMBL20628784

SCHEMBL20628784

C[C@H]1CC[C@@](C)(c2cc(NC(=O)c3nccn3C)ccc2F)N=C1N

nearest known ligand 0.61

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 12/20 0.61
BACE2 Q9Y5Z0 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4087666 0.83 BACE1 (0.68) BACE1BACE2
SCHEMBL4085379 0.83 BACE1 (0.68) BACE1BACE2
SCHEMBL20628895 0.81 BACE1 (0.75) BACE1BACE2
SCHEMBL20628563 0.81 BACE1 (0.66) BACE1BACE2
SCHEMBL12301647 0.79 BACE1 (0.60) BACE1BACE2
SCHEMBL20628958 0.79 BACE1 (0.69) BACE1BACE2
SCHEMBL20628779 0.79 BACE1 (0.70) BACE1BACE2
SCHEMBL20628730 0.78 BACE1 (0.69) BACE1BACE2
SCHEMBL20628777 0.78 BACE1 (0.74) BACE1BACE2
SCHEMBL20628930 0.78 BACE1 (0.72) BACE1BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3218362-B1 2-AMINO-3,5-DIFLUORO-3,6-DIMETHYL-6-PHENYL-3,4,5,6-TETRAHYDROPYRIDINES AS BACE1 INHIBITORS FOR TREATING ALZHEIMER'S DISEASE H LUNDBECK AS (DK) 2019-01-09 EP disclosed