SCHEMBL20631069

SCHEMBL20631069

On1cc(C(F)(F)F)c2sccc21

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.34
ADORA2A P29274 3/20 0.31
ADORA1 P30542 2/20 0.31
GAA P10253 2/20 0.30
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20673887 0.76 KMT2A (0.33)
SCHEMBL5174008 0.71 NTRK1 (0.32)
SCHEMBL20631042 0.71 GAA (0.32) GAA
SCHEMBL21958627 0.70 CA2 (0.34) CA2
SCHEMBL20674023 0.67 CA2 (0.41) CA2GAAKDM4EALDH1A1
SCHEMBL21955856 0.67 MEN1 (0.46) GAAALDH1A1
SCHEMBL20631034 0.67
SCHEMBL20631059 0.66 KDM4E (0.35) KDM4EALDH1A1
SCHEMBL21958543 0.66 CNOT7 (0.30) CA2
SCHEMBL20631027 0.66 FEN1 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019010295-A1 SELECTIVE INHIBITORS OF CLINICALLY IMPORTANT MUTANTS OF THE EGFR TYROSINE KINASE CS PHARMATECH LIMITED (KY) 2019-01-10 WO disclosed