SCHEMBL20633744

SCHEMBL20633744

O=c1c2ccccc2c2c(-c3ccccc3)cc(-c3ccccc3)cc2n1-c1cc(-c2ccccc2)cc(-c2ccc(-c3ccc4c(=O)n(-c5ccccc5)c5ccc6ncccc6c5c4c3)cc2)c1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ACVR1 Q04771 5/20 0.38
KMT2A Q03164 3/20 0.37
MEN1 O00255 2/20 0.37
HSP90AA1 P07900 1/20 0.37
MAPT P10636 1/20 0.37
PIK3CA P42336 1/20 0.36
ALDH1A1 P00352 3/20 0.35
CYP2C19 P33261 2/20 0.35
LOXL3 P58215 1/20 0.35
LOXL2 Q9Y4K0 1/20 0.35
TSHR P16473 1/20 0.35
EGLN1 Q9GZT9 1/20 0.34
CYP1A1 P04798 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP1B1 Q16678 1/20 0.34
PDE10A Q9Y233 1/20 0.33
MDM2 Q00987 1/20 0.32
GRK2 P25098 1/20 0.32
CYP2C9 P11712 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14933485 0.86 CYP1A1 (0.40) ACVR1KMT2AMEN1HSP90AA1MAPT
SCHEMBL14933580 0.80 MAPK1 (0.41) KMT2AMEN1HSP90AA1MAPTALDH1A1
SCHEMBL14933409 0.80 MAPK1 (0.49) ACVR1KMT2AMAPTALDH1A1CYP2C19
SCHEMBL13087158 0.74 ACVR1 (0.43) ACVR1KMT2AMEN1MAPTPIK3CA
SCHEMBL20633107 0.72 L3MBTL1 (0.45) KMT2AMEN1MAPTALDH1A1TSHR
SCHEMBL16483821 0.72 PIK3CA (0.39) ACVR1PIK3CAALDH1A1CYP2C19TSHR
SCHEMBL21636097 0.71 MAPK1 (0.47) KMT2AMEN1HSP90AA1MAPTALDH1A1
SCHEMBL15945619 0.71 KDM4E (0.46) ACVR1KMT2AMEN1MAPTPIK3CA
SCHEMBL16483579 0.71 PIK3CA (0.42) ACVR1PIK3CA
SCHEMBL25569981 0.71 L3MBTL1 (0.43) KMT2AMEN1HSP90AA1MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3649213-B1 COMPOSITION FOR ORGANIC ELECTRONIC DEVICES MERCK PATENT GMBH (DE) 2021-06-23 EP disclosed
WO-2019007867-A1 COMPOSITION FOR ORGANIC ELECTRONIC DEVICES MERCK PATENT GMBH (DE) 2019-01-10 WO disclosed