SCHEMBL20649338

SCHEMBL20649338

CC1(C)Cc2cnc(N)nc2-c2[nH]nc(C(=O)Nc3nc(CN4CCCC4)cs3)c21

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACKR3 P25106 2/20 0.36
DCPS Q96C86 1/20 0.35
CSNK2A1 P68400 1/20 0.35
CDK2 P24941 4/20 0.34
AURKA O14965 3/20 0.34
DYRK1A Q13627 2/20 0.34
CLK2 P49760 1/20 0.34
CLK3 P49761 1/20 0.34
BRPF1 P55201 1/20 0.33
ADRA2B P18089 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
TMEM97 Q5BJF2 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
GCK P35557 1/20 0.33
F2 P00734 2/20 0.33
F10 P00742 2/20 0.33
CCNA2 P20248 1/20 0.33
CCNA1 P78396 1/20 0.33
MAOB P27338 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20649227 0.93 DCPS (0.38) ACKR3DCPSCSNK2A1CDK2AURKA
SCHEMBL30183190 0.92 ACKR3 (0.36) ACKR3DCPSCSNK2A1CDK2AURKA
SCHEMBL20649082 0.92 ACKR3 (0.36) ACKR3DCPSCSNK2A1CDK2AURKA
Hydrochloric Acid SCHEMBL30183135 0.92 DCPS (0.38) ACKR3DCPSCSNK2A1CDK2AURKA
Hydrochloric Acid SCHEMBL21875647 0.92 DCPS (0.38) ACKR3DCPSCSNK2A1CDK2AURKA
SCHEMBL30183727 0.91 DCPS (0.37) ACKR3DCPSCSNK2A1CDK2AURKA
SCHEMBL20649269 0.91 DCPS (0.37) ACKR3DCPSCSNK2A1CDK2AURKA
SCHEMBL20649081 0.89 F2 (0.43) CSNK2A1F2F10MAOBAOC3
SCHEMBL20649045 0.89 CSNK2A1 (0.37) CSNK2A1CDK2GCKMAOBAOC3
SCHEMBL20649331 0.88 DCPS (0.35) ACKR3DCPSCSNK2A1CDK2AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019011715-A1 PYRAZOLO-QUINAZOLINE DERIVATIVES AS CHOLINE KINASE INHIBITORS NERVIANO MEDICAL SCIENCES S.R.L. (IT) 2019-01-17 WO disclosed