SCHEMBL20655868

SCHEMBL20655868

CC1(C)CCSc2ccc(C#Cc3ccc(C#N)nc3)cc21

nearest known ligand 0.65

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.65
CYP26A1 O43174 2/20 0.65
RARB P10826 10/20 0.59
RARG P13631 10/20 0.59
RARA P10276 9/20 0.59
KMT2A Q03164 1/20 0.59
CRABP2 P29373 1/20 0.36
BACE1 P56817 9/20 0.35
BACE2 Q9Y5Z0 9/20 0.35
RXRA P19793 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5485071 0.92 CYP3A4 (0.70) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL19342896 0.87 CYP3A4 (0.57) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL17885757 0.83 CYP3A4 (0.71) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL19034088 0.83 RARB (0.62) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL6665694 0.82 CYP3A4 (0.70) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL180442 0.81 CYP3A4 (0.70) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL30374281 0.80 CYP3A4 (0.69) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL860637 0.80 CYP3A4 (0.69) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL14330777 0.79 CYP3A4 (0.84) CYP3A4CYP26A1RARBRARGRARA
Tazarotenic Acid SCHEMBL678713 0.79 CYP3A4 (1.00) CYP3A4CYP26A1RARBRARGRARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3428155-A1 RETINOID COMPOUND, PREPARATION METHOD THEREFOR, INTERMEDIATES THEREOF AND APPLICATION THEREOF Shanghai Institute of Organic Chemistry, Chinese Academy of Sciences (CN) 2019-01-16 EP disclosed