SCHEMBL20659701

SCHEMBL20659701

COc1ccc(-c2cn(COCC[Si](C)(C)C)c3nccc(Oc4c(F)cc([N+](=O)[O-])cc4F)c23)cc1C#N

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TBK1 Q9UHD2 9/20 0.40
MAP4K1 Q92918 2/20 0.35
SCN9A Q15858 5/20 0.33
EGFR P00533 1/20 0.32
IGF1R P08069 1/20 0.32
SRC P12931 1/20 0.32
FLT4 P35916 1/20 0.32
KDR P35968 1/20 0.32
FLT3 P36888 1/20 0.32
EPHB4 P54760 1/20 0.32
TEK Q02763 1/20 0.32
KDM1A O60341 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29821698 1.00 TBK1 (0.40) TBK1MAP4K1SCN9AEGFRIGF1R
SCHEMBL29822161 0.93 TBK1 (0.33) TBK1MAP4K1SCN9A
SCHEMBL29822168 0.92 TBK1 (0.43) TBK1MAP4K1
SCHEMBL20659189 0.92 TBK1 (0.43) TBK1MAP4K1
SCHEMBL20659048 0.92 TBK1 (0.43) TBK1MAP4K1
SCHEMBL29821475 0.92 TBK1 (0.43) TBK1MAP4K1
SCHEMBL20659000 0.91 TBK1 (0.34) TBK1MAP4K1EGFRIGF1RSRC
SCHEMBL29821892 0.91 TBK1 (0.34) TBK1MAP4K1EGFRIGF1RSRC
SCHEMBL20659343 0.89 ALOX5AP (0.31)
SCHEMBL29822307 0.89 ALOX5AP (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3655406-A1 SUBSTITUTED PYRROLOPYRIDINE-DERIVATIVES Bayer Pharma Aktiengesellschaft (DE) 2020-05-27 EP disclosed
WO-2019016071-A1 SUBSTITUTED PYRROLOPYRIDINE-DERIVATIVES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2019-01-24 WO disclosed