SCHEMBL20688147

SCHEMBL20688147

CNc1cccn([C@@H]2CCN(C)C[C@@H]2F)c1=O

nearest known ligand 0.52

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
TYK2 P29597 20/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21227384 1.00 TYK2 (0.52) TYK2
SCHEMBL20688144 1.00 TYK2 (0.52) TYK2
SCHEMBL21227385 1.00 TYK2 (0.52) TYK2
SCHEMBL20696760 0.86 TYK2 (0.45) TYK2
SCHEMBL20696762 0.86 TYK2 (0.45) TYK2
SCHEMBL21227388 0.86 TYK2 (0.45) TYK2
SCHEMBL21285356 0.86 TYK2 (0.45) TYK2
SCHEMBL24880689 0.83 TYK2 (0.45) TYK2
SCHEMBL21227516 0.83 TYK2 (0.45) TYK2
SCHEMBL20689432 0.81 TYK2 (0.40) TYK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020154474-A1 TYK2 INHIBITORS AND USES THEREOF NIMBUS LAKSHMI, INC. (US) 2020-07-30 WO disclosed
WO-2019023468-A1 TYK2 INHIBITORS AND USES THEREOF NIMBUS LAKSHMI, INC. (US) 2019-01-31 WO disclosed