SCHEMBL20713634

SCHEMBL20713634

CNC(=O)CNC(=O)c1csc(C2CCCN2C(=O)c2cn(C)c(C)n2)n1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 7/20 0.43
TRPC3 Q13507 3/20 0.37
TRPC6 Q9Y210 3/20 0.37
TRPV1 Q8NER1 4/20 0.35
TRPA1 O75762 1/20 0.35
CACNA1C Q13936 1/20 0.35
SCN5A Q14524 1/20 0.35
TRPV4 Q9HBA0 1/20 0.35
BAZ2A Q9UIF9 1/20 0.35
ACKR3 P25106 1/20 0.35
NAA50 Q9GZZ1 1/20 0.34
FAP Q12884 1/20 0.33
HSD11B1 P28845 1/20 0.32
CPT2 P23786 1/20 0.32
CPT1A P50416 1/20 0.32
CPT1B Q92523 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20713640 0.84 KLKB1 (0.55) KLKB1TRPC3TRPC6
SCHEMBL20713726 0.83 BAZ2A (0.43) KLKB1TRPC3TRPC6TRPV1TRPA1
SCHEMBL20713811 0.83 TRPC3 (0.43) KLKB1TRPC3TRPC6TRPV1TRPA1
SCHEMBL20713814 0.83 TRPC3 (0.43) KLKB1TRPC3TRPC6TRPV1TRPA1
SCHEMBL20713771 0.83 TRPC3 (0.42) KLKB1TRPC3TRPC6TRPV1ACKR3
SCHEMBL20713774 0.83 ACKR3 (0.44) KLKB1TRPV1BAZ2AACKR3NAA50
SCHEMBL20713724 0.82 KLKB1 (0.51) KLKB1
SCHEMBL20713642 0.81 KLKB1 (0.40) KLKB1TRPV1BAZ2AACKR3NAA50
SCHEMBL20713881 0.81 KLKB1 (0.38) KLKB1TRPV1BAZ2AACKR3NAA50
SCHEMBL20713770 0.81 SMN1; SMN2 (0.44) KLKB1TRPC3TRPC6BAZ2AHSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019028362-A1 INHIBITORS OF PLASMA KALLIKREIN AND USES THEREOF DYAX CORP. (US) 2019-02-07 WO disclosed