SCHEMBL2071769

SCHEMBL2071769

CC(C)C(C(=O)O)n1nnnc1N1CCC(NC(=O)c2ccc(-c3cccc(F)c3)nc2)CC1

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 9/20 0.57
ALDH1A1 P00352 1/20 0.43
POLB P06746 1/20 0.43
USP30 Q70CQ3 1/20 0.43
MAP4K4 O95819 1/20 0.41
CYP2C9 P11712 4/20 0.40
MAPK14 Q16539 4/20 0.40
GABRA5 P31644 2/20 0.40
SMO Q99835 1/20 0.40
DRD2 P14416 1/20 0.40
DRD4 P21917 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2071903 0.91 HPGDS (0.61) HPGDSALDH1A1POLBUSP30MAP4K4
SCHEMBL2073136 0.90 HPGDS (0.57) HPGDSALDH1A1POLBUSP30MAP4K4
SCHEMBL2073082 0.86 HPGDS (0.57) HPGDSALDH1A1POLBUSP30GABRA5
SCHEMBL2070062 0.86 HPGDS (0.63) HPGDSALDH1A1POLBUSP30MAP4K4
SCHEMBL2070308 0.84 HPGDS (0.60) HPGDSALDH1A1POLBUSP30DRD2
SCHEMBL5061048 0.83 HPGDS (0.61) HPGDSALDH1A1POLBUSP30MAP4K4
SCHEMBL2073193 0.82 HPGDS (0.57) HPGDSALDH1A1POLBUSP30MAP4K4
SCHEMBL2071036 0.82 HPGDS (0.61) HPGDSALDH1A1POLBUSP30MAP4K4
SCHEMBL2070154 0.81 HPGDS (0.58) HPGDSALDH1A1POLBUSP30MAP4K4
SCHEMBL2071686 0.79 HPGDS (0.65) HPGDSUSP30GABRA5DRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7902373-B2 asthma; for treating prostaglandin D2 mediated diseases; e.g. 6-(3-fluorophenyl)-N-[1-(1-methyl-1H-tetrazol-5-yl)piperidin-4-yl]nicotinamide PFIZER INC (US) 2011-03-08 US disclosed