SCHEMBL2072154

SCHEMBL2072154

CN1CC[C@H](Oc2cc(Oc3ccc(C(=O)N4CCC4)cc3)cc(C(=O)Nc3ccn(C(=O)O)n3)c2)C1=O

nearest known ligand 0.62

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
GCK P35557 20/20 0.62
KCNH2 Q12809 11/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2657684 0.90 GCK (0.58) GCKKCNH2
SCHEMBL2072152 0.90 GCK (0.58) GCKKCNH2
SCHEMBL2073632 0.86 GCK (0.56) GCKKCNH2
SCHEMBL2657879 0.84 GCK (0.65) GCKKCNH2
SCHEMBL2074921 0.84 GCK (0.65) GCKKCNH2
SCHEMBL2074591 0.82 GCK (0.48) GCKKCNH2
SCHEMBL2657926 0.80 GCK (0.49) GCKKCNH2
SCHEMBL2072002 0.80 GCK (0.49) GCKKCNH2
SCHEMBL2074125 0.80 GCK (0.43) GCKKCNH2
SCHEMBL2653806 0.79 GCK (0.87) GCKKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7902200-B2 3-[6-(Azetidine-1-carbonyl)pyridin-3-yl]oxy-5-[(3S)-1-methyl-2-oxo-pyrrolidin-3-yl]oxy-N-(5-methylpyrazin-2-yl)benzamide; activates glucokinase leading to decreased glucose threshold for insulin secretion and lowering of blood glucose by increasing hepatic glucose uptake; antidiabetic agents; obesity ASTRAZENECA AB (SE) 2011-03-08 US disclosed
US-20080171734-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2008-07-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080171734-A1 CHEMICAL COMPOUNDS HK1, GCKR, GCK GCK 3/4885KCNH2 1008/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.