SCHEMBL20729439

SCHEMBL20729439

O[C@H]1CCN(CCCOS)C1

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 12/20 0.49
HRH2 P25021 4/20 0.49
HRH1 P35367 4/20 0.49
PDCD1 Q15116 1/20 0.44
CD274 Q9NZQ7 1/20 0.44
HTR1A P08908 1/20 0.43
LTA4H P09960 1/20 0.41
ACHE P22303 1/20 0.38
PDK2 Q15119 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24114470 1.00 HRH3 (0.49) HRH3HRH2HRH1PDCD1CD274
SCHEMBL20729442 0.89 HTR1A (0.55) HRH3HRH2HRH1PDCD1CD274
SCHEMBL20729454 0.89 HRH3 (0.47) HRH3HRH2HRH1ACHE
SCHEMBL28960041 0.82 PDCD1 (0.49) HRH3HRH2HRH1PDCD1CD274
SCHEMBL13552419 0.81 HRH3 (0.49) HRH3HRH2HRH1PDCD1CD274
SCHEMBL12717290 0.81 HRH3 (0.49) HRH3HRH2HRH1PDCD1CD274
SCHEMBL9921265 0.81 HRH3 (0.49) HRH3HRH2HRH1PDCD1CD274
SCHEMBL10059171 0.80 HRH3 (0.48) HRH3HRH2HRH1PDCD1CD274
SCHEMBL10059156 0.80 HRH3 (0.48) HRH3HRH2HRH1PDCD1CD274
SCHEMBL21310147 0.80 HRH3 (0.34) HRH3HRH2HRH1HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019165043-A2 INDANE-AMINES AS PD-L1 ANTAGONISTS CHEMOCENTRYX, INC. (US) 2019-08-29 WO disclosed
WO-2019032547-A1 MACROCYCLIC IMMUNOMODULATORS CHEMOCENTRYX, INC. (US) 2019-02-14 WO disclosed