SCHEMBL20729848

SCHEMBL20729848

O=C(O)NCCNC(=S)Nc1ccc2c(c1)C(=O)OC21c2ccc(O)cc2Oc2cc(O)ccc21

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FTO Q9C0B1 8/20 0.66
NAALAD2 Q9Y3Q0 4/20 0.60
TTR P02766 1/20 0.59
KEAP1 Q14145 1/20 0.54
JAK2 O60674 1/20 0.53
MEN1 O00255 1/20 0.53
MAPT P10636 1/20 0.53
HPGD P15428 1/20 0.53
CYP2C19 P33261 1/20 0.53
HTT P42858 1/20 0.53
RECQL P46063 1/20 0.53
BLM P54132 1/20 0.53
SMAD3 P84022 1/20 0.53
KMT2A Q03164 1/20 0.53
PRMT1 Q99873 1/20 0.53
ACE2 Q9BYF1 1/20 0.53
TDP1 Q9NUW8 1/20 0.53
NQO1 P15559 1/20 0.52
DRD1 P21728 1/20 0.52
MAP1LC3B Q9GZQ8 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12754623 0.91 FTO (0.65) FTONAALAD2TTRKEAP1JAK2
SCHEMBL17037385 0.90 FTO (0.66) FTONAALAD2TTRKEAP1JAK2
SCHEMBL17956697 0.90 FTO (0.69) FTONAALAD2TTRKEAP1JAK2
SCHEMBL18461840 0.90 FTO (0.77) FTONAALAD2TTRKEAP1JAK2
SCHEMBL20729847 0.90 FTO (0.66) FTONAALAD2TTRKEAP1JAK2
SCHEMBL17589330 0.89 FTO (0.64) FTONAALAD2TTRKEAP1JAK2
SCHEMBL29368721 0.89 FTO (0.64) FTONAALAD2TTRKEAP1JAK2
SCHEMBL9293647 0.89 FTO (0.64) FTONAALAD2TTRKEAP1JAK2
SCHEMBL22863319 0.89 NAALAD2 (0.63) FTONAALAD2TTRKEAP1JAK2
SCHEMBL20809317 0.89 FTO (0.70) FTONAALAD2TTRKEAP1JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3665161-B1 NEW TARGETED CYTOTOXIC RATJADONE DERIVATIVES AND CONJUGATES THEREOF HELMHOLTZ ZENTRUM INFEKTIONSFORSCHUNG GMBH (DE) 2023-09-27 EP disclosed
WO-2019030284-A1 NEW TARGETED CYTOTOXIC RATJADONE DERIVATIVES AND CONJUGATES THEREOF Helmholtz-Zentrum für Infektionsforschung GmbH (DE) 2019-02-14 WO disclosed