SCHEMBL20734937

SCHEMBL20734937

CC(C)(C)OC(=O)N1C(=O)C=C(OCCc2ccccn2)C1Cc1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KLK7 P49862 8/20 0.46
KLK5 Q9Y337 7/20 0.43
PRSS1 P07477 3/20 0.42
PRSS2 P07478 3/20 0.42
PRSS3 P35030 3/20 0.42
KDM4E B2RXH2 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
PLA2G10 O15496 1/20 0.36
PLA2G5 P39877 1/20 0.36
CYP3A4 P08684 1/20 0.36
ALOX15 P16050 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
CYP1A2 P05177 1/20 0.35
GPR119 Q8TDV5 1/20 0.35
TAAR1 Q96RJ0 1/20 0.35
PDE10A Q9Y233 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20734936 1.00 KLK7 (0.46) KLK7KLK5PRSS1PRSS2PRSS3
SCHEMBL20735102 0.89 KLK7 (0.52) KLK7KLK5PRSS1PRSS2PRSS3
SCHEMBL20735103 0.89 KLK7 (0.52) KLK7KLK5PRSS1PRSS2PRSS3
SCHEMBL20734892 0.83 KLK7 (0.51) KLK7KLK5PRSS1PRSS2PRSS3
SCHEMBL20734894 0.83 KLK7 (0.51) KLK7KLK5PRSS1PRSS2PRSS3
SCHEMBL20735107 0.83 KLK7 (0.57) KLK7KLK5PRSS1PRSS2PRSS3
SCHEMBL20735106 0.83 KLK7 (0.57) KLK7KLK5PRSS1PRSS2PRSS3
SCHEMBL20734817 0.79 KLK7 (0.47) KLK7KLK5PRSS1PRSS2PRSS3
SCHEMBL20734818 0.79 KLK7 (0.47) KLK7KLK5PRSS1PRSS2PRSS3
SCHEMBL20734886 0.79 KLK7 (0.48) KLK7KLK5PRSS1PRSS2PRSS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019029273-A1 4-OXO-ALKYLATED TETRAMIC ACID COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF 北京卓凯生物技术有限公司 2019-02-14 WO disclosed
WO-2019029274-A1 4-OXO-ALKYLATED TETRAMIC ACID COMPOUND AND PREPARATION METHOD THEREFOR 北京卓凯生物技术有限公司 2019-02-14 WO disclosed