SCHEMBL20748852

SCHEMBL20748852

Cc1nn2c(c1C(N)=O)CB(C#N)CC2

nearest known ligand 0.31

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CSNK1D P48730 2/20 0.31
CSNK1E P49674 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20748843 0.88 POLB (0.31)
SCHEMBL20748874 0.82 PDE4D (0.36)
SCHEMBL20748885 0.78 CSNK1E (0.48) CSNK1DCSNK1E
SCHEMBL21131229 0.77 CSNK1E (0.51) CSNK1DCSNK1E
SCHEMBL20748882 0.76 CSNK1E (0.46) CSNK1DCSNK1E
SCHEMBL20748938 0.74 RIPK2 (0.45) CSNK1DCSNK1E
SCHEMBL20748937 0.74 CSNK1E (0.52) CSNK1DCSNK1E
SCHEMBL20748866 0.74 CSNK1E (0.55) CSNK1DCSNK1E
SCHEMBL20748869 0.71
SCHEMBL20748895 0.67 TLR9 (0.42) CSNK1DCSNK1E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3068785-B1 SUBSTITUTED 4,5,6,7-TETRAHYDROPYRAZOLO[1,5-A]PYRAZINE DERIVATIVES AS CASEIN KINASE 1 D/E INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2019-06-26 EP disclosed
EP-3068784-B1 SUBSTITUTED 4,5,6,7-TETRAHYDROPYRAZOLO[1,5-A]PYRAZINE DERIVATIVES AS CASEIN KINASE 1 D/E INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2019-02-20 EP disclosed