SCHEMBL20763538

SCHEMBL20763538

COc1nc(OCc2cccc(COc3ccc(CNCCNC(C)=O)c(OC)n3)c2C)ccc1CNCCNC(C)=O

nearest known ligand 0.90

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CD274 Q9NZQ7 19/20 0.90
PDCD1 Q15116 15/20 0.90
PDCD1LG2 Q9BQ51 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30574115 0.95 CD274 (1.00) CD274PDCD1PDCD1LG2
SCHEMBL19849668 0.95 CD274 (1.00) CD274PDCD1PDCD1LG2
SCHEMBL20763763 0.91 CD274 (0.93) CD274PDCD1PDCD1LG2
SCHEMBL22132095 0.91 CD274 (0.93) CD274PDCD1PDCD1LG2
SCHEMBL20763743 0.91 CD274 (0.75) CD274PDCD1PDCD1LG2
SCHEMBL20763755 0.91 CD274 (0.75) CD274PDCD1PDCD1LG2
SCHEMBL16566296 0.91 CD274 (1.00) CD274PDCD1
SCHEMBL29382060 0.91 CD274 (1.00) CD274PDCD1
Hydrochloric Acid SCHEMBL19100243 0.90 CD274 (1.00) CD274PDCD1
SCHEMBL20763783 0.90 CD274 (0.89) CD274PDCD1PDCD1LG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11787766-B2 Compound having PD-L1 inhibitory activity, preparation method therefor and use thereof SHANGHAI ENNOVABIO PHARMACEUTICALS CO., LTD. (CN) 2023-10-17 US disclosed
US-20200392083-A1 COMPOUND HAVING PD-L1 INHIBITORY ACTIVITY, PREPARATION METHOD THEREFOR AND USE THEREOF SHANGHAI ENNOVABIO PHARMACEUTICALS CO., LTD. (CN) 2020-12-17 US disclosed
EP-3669872-A1 COMPOUND HAVING PD-L1 INHIBITORY ACTIVITY, PREPARATION METHOD THEREFOR AND USE THEREOF Shanghai Ennovabio Pharmaceuticals Co., Ltd. (CN) 2020-06-24 EP disclosed
WO-2019034172-A1 COMPOUND HAVING PD-L1 INHIBITORY ACTIVITY, PREPARATION METHOD THEREFOR AND USE THEREOF 上海轶诺药业有限公司 2019-02-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200392083-A1 COMPOUND HAVING PD-L1 INHIBITORY ACTIVITY, PREPARATION METHOD THEREFOR AND USE THEREOF CD274, PDCD1LG2, PDCD1 CD274 1/4885PDCD1 3/4885PDCD1LG2 2/4885
US-11787766-B2 Compound having PD-L1 inhibitory activity, preparation method therefor and use thereof CD274, PDCD1, PDCD1LG2 CD274 1/4885PDCD1 2/4885PDCD1LG2 3/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.