SCHEMBL20765633

SCHEMBL20765633

O=C(CCc1ccccc1)N1CCN(C(=O)c2ccc3cc[nH]c3c2)CC1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 3/20 0.71
GHSR Q92847 4/20 0.67
NPC1 O15118 2/20 0.52
TDP1 Q9NUW8 1/20 0.52
KDM4E B2RXH2 3/20 0.52
POLB P06746 3/20 0.52
MAPK1 P28482 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
FKBP1A P62942 1/20 0.49
TSHR P16473 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
ALDH1A1 P00352 2/20 0.48
HPGD P15428 1/20 0.48
ENPP2 Q13822 1/20 0.48
HSD17B10 Q99714 1/20 0.48
MAPT P10636 1/20 0.47
ME2 P23368 1/20 0.47
ME1 P48163 1/20 0.47
ME3 Q16798 1/20 0.47
GFER P55789 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6095301 0.86 MAPK14 (0.79) MAPK14GHSRNPC1KDM4EALDH1A1
SCHEMBL20765535 0.81 KDM4E (0.57) MAPK14NPC1TDP1KDM4EPOLB
SCHEMBL20765688 0.81 GHSR (0.65) MAPK14GHSRNPC1POLBSMN1; SMN2
SCHEMBL20765500 0.81 MAPK14 (0.70) MAPK14GHSRNPC1KDM4EMAPK1
SCHEMBL14028477 0.80 GHSR (1.00) MAPK14GHSRMAPK1HPGD
SCHEMBL17443852 0.80 GHSR (0.75) MAPK14GHSRKDM4EALDH1A1HPGD
SCHEMBL6093708 0.78 MAPK14 (0.79) MAPK14GHSRNPC1
SCHEMBL27158221 0.77 MAPK14 (0.65) MAPK14GHSRKDM4EALDH1A1HPGD
SCHEMBL7131839 0.76 NPC1 (0.86) NPC1TDP1POLBSMN1; SMN2FKBP1A
SCHEMBL16598935 0.76 GHSR (0.70) MAPK14GHSRKDM4ESMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019038683-A1 COMPOUNDS TARGETING TANDEM BRCT DOMAINS OF BRCA1, COMPOSITIONS AND METHODS THEREOF INSTITUTE FOR STEM CELL BIOLOGY AND REGENERATIVE MEDICINE (IN) 2019-02-28 WO claimed