SCHEMBL2076570

SCHEMBL2076570

O=C(Nc1cc(N2CCN(C3CCCC3)CC2)ncn1)N1CCC(C(F)(F)F)CC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.50
PDGFRB P09619 1/20 0.43
SMN1; SMN2 Q16637 3/20 0.41
ALDH1A1 P00352 3/20 0.41
RAB9A P51151 2/20 0.41
DRD2 P14416 1/20 0.39
DRD3 P35462 1/20 0.39
AXL P30530 1/20 0.39
MERTK Q12866 1/20 0.39
EGFR P00533 1/20 0.38
ERBB3 P21860 1/20 0.38
FAAH O00519 1/20 0.37
CNR2 P34972 1/20 0.37
P4HTM Q9NXG6 1/20 0.37
KDM4E B2RXH2 1/20 0.37
GAA P10253 1/20 0.37
HTT P42858 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
NPC1 O15118 1/20 0.37
ATM Q13315 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2075465 0.99 HRH4 (0.52) HRH4PDGFRBSMN1; SMN2ALDH1A1RAB9A
SCHEMBL2075851 0.89 HRH4 (0.51) HRH4PDGFRBSMN1; SMN2ALDH1A1RAB9A
SCHEMBL2074092 0.89 HRH4 (0.53) HRH4PDGFRBSMN1; SMN2ALDH1A1RAB9A
SCHEMBL2076138 0.88 HRH4 (0.54) HRH4PDGFRBSMN1; SMN2ALDH1A1RAB9A
SCHEMBL2074954 0.87 HRH4 (0.55) HRH4PDGFRBSMN1; SMN2ALDH1A1RAB9A
SCHEMBL2074480 0.87 HRH4 (0.55) HRH4PDGFRBSMN1; SMN2ALDH1A1RAB9A
SCHEMBL2075259 0.87 HRH4 (0.55) HRH4PDGFRBSMN1; SMN2ALDH1A1RAB9A
SCHEMBL2074889 0.87 HRH4 (0.55) HRH4PDGFRBSMN1; SMN2ALDH1A1RAB9A
SCHEMBL2074972 0.87 HRH4 (0.55) HRH4PDGFRBSMN1; SMN2ALDH1A1RAB9A
SCHEMBL2074130 0.86 HRH4 (0.53) HRH4PDGFRBSMN1; SMN2ALDH1A1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7902184-B2 Piperazinyl pyrimidine derivatives HOFFMANN-LA ROCHE INC. (US) 2011-03-08 US disclosed