SCHEMBL20766653

SCHEMBL20766653

O=C1NCCCCC1N1Cc2c(O)cccc2C1=O

nearest known ligand 0.64

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 6/20 0.64
IKZF3 Q9UKT9 2/20 0.47
IKZF1 Q13422 2/20 0.47
BRD4 O60885 1/20 0.47
TNF P01375 1/20 0.47
IL1B P01584 1/20 0.47
DDB1 Q16531 1/20 0.47
MAP1LC3B Q9GZQ8 11/20 0.44
PARP1 P09874 1/20 0.40
CSNK1A1 P48729 1/20 0.39
CDK5 Q00535 1/20 0.39
DYRK1A Q13627 1/20 0.39
CDK5R1 Q15078 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20766651 1.00 CRBN (0.64) CRBNIKZF3IKZF1BRD4TNF
SCHEMBL19611961 0.86 CRBN (0.47) CRBNIKZF3IKZF1BRD4TNF
SCHEMBL19611971 0.86 CRBN (0.50) CRBNIKZF3IKZF1BRD4TNF
SCHEMBL19612062 0.86 HTR2A (0.48) CRBNIKZF3IKZF1BRD4TNF
SCHEMBL19611910 0.86 MAPK1 (0.53) CRBNIKZF3IKZF1BRD4TNF
SCHEMBL19612063 0.86 HTR2A (0.48) CRBNIKZF3IKZF1BRD4TNF
SCHEMBL18270984 0.86 HTR2A (0.48) CRBNIKZF3IKZF1BRD4TNF
SCHEMBL19611973 0.86 CRBN (0.50) CRBNIKZF3IKZF1BRD4TNF
SCHEMBL19611911 0.86 MAPK1 (0.53) CRBNIKZF3IKZF1BRD4TNF
SCHEMBL18263930 0.86 CRBN (0.65) CRBNIKZF3IKZF1BRD4TNF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10927104-B2 Ether compounds and uses thereof BIOTHERYX, INC. (US) 2021-02-23 US disclosed
US-20200231582-A1 ETHER COMPOUNDS AND USES THEREOF BIOTHERYX, INC. 2020-07-23 US disclosed
EP-3672955-A1 ETHER COMPOUNDS AND USES THEREOF Biotheryx Inc. (US) 2020-07-01 EP disclosed
CN-111247138-A Ether compound and use thereof 拜欧赛里克斯公司 2020-06-05 CN disclosed
WO-2019040274-A1 ETHER COMPOUNDS AND USES THEREOF BIOTHERYX, INC. (US) 2019-02-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10927104-B2 Ether compounds and uses thereof EPCAM, ICAM1, SELE CRBN 379/4885IKZF3 122/4885IKZF1 343/4885
US-20200231582-A1 ETHER COMPOUNDS AND USES THEREOF EPCAM, ICAM1, SELE CRBN 379/4885IKZF3 122/4885IKZF1 343/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.