SCHEMBL20780841

SCHEMBL20780841

CNc1ccc2ncnc(Nc3ccc(Oc4ccc5nc[nH]c5c4)c(C)c3)c2c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAF1 P04049 1/20 0.52
BRAF P15056 1/20 0.52
ERBB2 P04626 12/20 0.51
EGFR P00533 11/20 0.51
ERBB3 P21860 2/20 0.50
ERBB4 Q15303 2/20 0.50
FECH P22830 2/20 0.47
NQO2 P16083 1/20 0.47
MYH14 Q7Z406 1/20 0.47
RIPK3 Q9Y572 1/20 0.47
MAPT P10636 2/20 0.46
LMNA P02545 1/20 0.46
HTT P42858 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
CDK8 P49336 1/20 0.45
MAP2K5 Q13163 1/20 0.45
CDK19 Q9BWU1 1/20 0.45
MKNK2 Q9HBH9 1/20 0.45
NCOA1 Q15788 1/20 0.44
NCOA3 Q9Y6Q9 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22200858 0.85 EGFR (0.61) ERBB2EGFRERBB4
SCHEMBL12872982 0.80 ERBB2 (0.54) RAF1BRAFERBB2EGFRERBB3
SCHEMBL22076856 0.78 EGFR (0.47) ERBB2EGFRFECHCDK8MAP2K5
SCHEMBL15431012 0.78 ERBB2 (0.46) RAF1BRAFERBB2EGFRERBB3
SCHEMBL20780984 0.77 ERBB2 (0.59) ERBB2EGFRERBB3ERBB4FECH
SCHEMBL29025871 0.77 EGFR (0.68) ERBB2EGFR
SCHEMBL20780840 0.77 EGFR (0.68) ERBB2EGFR
SCHEMBL24832693 0.75 ERBB2 (0.68) ERBB2EGFRERBB3ERBB4FECH
SCHEMBL24569983 0.75 HTT (0.62) ERBB2EGFRERBB3ERBB4FECH
SCHEMBL24569330 0.74 ERBB2 (0.67) ERBB2EGFRERBB3ERBB4FECH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019042409-A1 NITROGENOUS HETEROCYCLIC COMPOUND, PREPARATION METHOD, INTERMEDIATE, COMPOSITION, AND APPLICATION 上海医药集团股份有限公司 2019-03-07 WO disclosed