SCHEMBL20782877

SCHEMBL20782877

COc1cc2ncnc(OC(C)C)c2cc1OC

nearest known ligand 0.57

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LCK P06239 2/20 0.57
SRC P12931 2/20 0.57
TRPA1 O75762 1/20 0.54
KDR P35968 7/20 0.51
EGFR P00533 6/20 0.51
RET P07949 2/20 0.51
KIF5B P33176 1/20 0.51
KRAS P01116 1/20 0.48
SOS1 Q07889 1/20 0.48
ENPP1 P22413 4/20 0.48
PDGFRA P16234 1/20 0.46
PDE1B Q01064 1/20 0.46
FLT3 P36888 1/20 0.46
GAK O14976 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1985538 0.84 LCK (0.66) LCKSRCTRPA1KDREGFR
SCHEMBL3332968 0.81 PIK3CA (0.57) TRPA1EGFRGAK
SCHEMBL13918286 0.80 ENPP1 (0.67) LCKSRCKDREGFRKRAS
SCHEMBL12003599 0.80 ENPP1 (0.67) LCKSRCKDREGFRKRAS
SCHEMBL13906935 0.79 LCK (0.60) LCKSRCTRPA1KDREGFR
SCHEMBL13757489 0.78 TRPA1 (0.56) LCKSRCTRPA1EGFRFLT3
SCHEMBL25671083 0.77 SRC (0.51) LCKSRCKDREGFRRET
SCHEMBL11316949 0.76 PDE1B (0.58) LCKSRCKDREGFRRET
SCHEMBL23457663 0.73 LCK (0.74) LCKTRPA1KDREGFRRET
SCHEMBL28891487 0.73 KIT (0.39) LCKSRCTRPA1KDREGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019046778-A1 ECTONUCLEOTIDE PYROPHOSPHATASE-PHOSPHODIESTERASE 1 (ENPP-1) INHIBITORS AND USES THEREOF MAVUPHARMA, INC. (US) 2019-03-07 WO disclosed