SCHEMBL20808262

SCHEMBL20808262

COc1cc(OC)c(F)c(N(Cc2nccn2SN(C)C)c2cc3cc(-c4cnn(C)c4)cnc3cn2)c1F

nearest known ligand 0.75

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
FGFR4 P22455 20/20 0.75
FGFR3 P22607 20/20 0.75
FGFR1 P11362 19/20 0.75
FGFR2 P21802 19/20 0.75
KDR P35968 13/20 0.75

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20808261 0.89 FGFR4 (0.76) FGFR4FGFR3FGFR1FGFR2KDR
SCHEMBL20808259 0.88 FGFR1 (0.75) FGFR4FGFR3FGFR1FGFR2KDR
SCHEMBL14905320 0.85 FGFR1 (1.00) FGFR4FGFR3FGFR1FGFR2KDR
SCHEMBL20808364 0.85 FGFR4 (0.74) FGFR4FGFR3FGFR1FGFR2KDR
SCHEMBL20808384 0.84 FGFR4 (0.66) FGFR4FGFR3FGFR1FGFR2KDR
SCHEMBL21128376 0.81 FGFR1 (0.65) FGFR4FGFR3FGFR1FGFR2KDR
SCHEMBL14905329 0.81 FGFR1 (1.00) FGFR4FGFR3FGFR1FGFR2KDR
SCHEMBL14905209 0.79 FGFR4 (1.00) FGFR4FGFR3FGFR1FGFR2KDR
SCHEMBL20808369 0.79 FGFR1 (0.75) FGFR4FGFR3FGFR1FGFR2KDR
SCHEMBL20808255 0.77 FGFR1 (0.74) FGFR4FGFR3FGFR1FGFR2KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2776436-B1 NEW COMPOUNDS ASTEX THERAPEUTICS LTD (GB) 2019-03-13 EP disclosed