SCHEMBL20835008

SCHEMBL20835008

CCCCc1ccc(C#Cc2cc(F)c(N=C=S)c(F)c2)c(CC)c1F

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 1/20 0.34
GABRB2 P47870 1/20 0.34
TYR P14679 1/20 0.33
FFAR1 O14842 1/20 0.31
FFAR4 Q5NUL3 1/20 0.31
MTNR1A P48039 1/20 0.30
MTNR1B P49286 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23309987 0.97 TYR (0.34) GABRA1GABRB2TYRFFAR1FFAR4
SCHEMBL23310000 0.93 GABRA1 (0.35) GABRA1GABRB2FFAR1FFAR4
SCHEMBL20835009 0.91 FFAR1 (0.33) GABRA1GABRB2TYRFFAR1FFAR4
SCHEMBL20834698 0.89 GABRA1 (0.41) GABRA1GABRB2FFAR1FFAR4
SCHEMBL20834947 0.86 TYR (0.32) TYRMTNR1AMTNR1B
SCHEMBL20834870 0.84 TYR (0.30) TYR
SCHEMBL28912870 0.84 FFAR1 (0.33) GABRA1GABRB2TYRFFAR1FFAR4
SCHEMBL20834945 0.83 MEN1 (0.32) TYRMTNR1AMTNR1B
SCHEMBL20834891 0.82 GABRA1 (0.37) GABRA1GABRB2FFAR1FFAR4MTNR1A
SCHEMBL20834901 0.81 MEN1 (0.31) TYR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3681976-B1 ISOTHIOCYANATO TOLANE DERIVATIVES MERCK PATENT GMBH (DE) 2021-05-26 EP disclosed
US-20210122977-A1 ISOTHIOCYANATO TOLANE DERIVATIVES MERCK PATENT GMBH (DE) 2021-04-29 US disclosed
WO-2019052972-A1 ISOTHIOCYANATO TOLANE DERIVATIVES MERCK PATENT GMBH (DE) 2019-03-21 WO disclosed