SCHEMBL20839717

SCHEMBL20839717

CCOC(=O)CCc1cccc(NC(=O)c2cc(OC)ccc2NC(=O)c2ccc3ccccc3c2)c1

nearest known ligand 0.70

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 7/20 0.70
PPARD Q03181 4/20 0.55
PPARG P37231 3/20 0.54
PPARA Q07869 3/20 0.54
NPC1 O15118 3/20 0.49
RAB9A P51151 3/20 0.49
CASP3 P42574 1/20 0.49
SENP7 Q9BQF6 1/20 0.49
F10 P00742 1/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
MAPT P10636 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
PLAU P00749 1/20 0.46
ABCG2 Q9UNQ0 1/20 0.46
RXFP1 Q9HBX9 1/20 0.46
KCNK3 O14649 1/20 0.45
KCNK9 Q9NPC2 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20839675 0.93 NR1H4 (0.81) NR1H4PPARDPPARGPPARANPC1
SCHEMBL20840618 0.91 NR1H4 (0.59) NR1H4PPARDPPARGPPARANPC1
SCHEMBL20839747 0.90 NR1H4 (0.58) NR1H4PPARDPPARGPPARANPC1
SCHEMBL20839666 0.89 NR1H4 (0.86) NR1H4PPARDPPARGPPARANPC1
SCHEMBL20839988 0.86 NR1H4 (0.67) NR1H4PPARDPPARGPPARANPC1
SCHEMBL20839936 0.84 NR1H4 (0.65) NR1H4PPARDPPARGPPARANPC1
SCHEMBL20839595 0.83 NR1H4 (0.66) NR1H4PPARDPPARGPPARANPC1
SCHEMBL20839731 0.83 NR1H4 (0.80) NR1H4PPARDPPARGPPARAMAPT
SCHEMBL20839500 0.82 NR1H4 (1.00) NR1H4PPARDPPARGPPARANPC1
SCHEMBL20839944 0.81 NR1H4 (0.49) NR1H4PPARDNPC1RAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019057969-A1 DUAL AGONISTS OF FXR AND PPARδ AND THEIR USES Johann Wolfgang Goethe-Universität (DE) 2019-03-28 WO disclosed