SCHEMBL20839747

SCHEMBL20839747

CCOC(=O)CCc1cccc(NC(=O)c2cc(Cl)ccc2NC(=O)c2ccc3ccccc3c2)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 8/20 0.58
HSPH1 Q92598 1/20 0.57
F10 P00742 2/20 0.57
PPARD Q03181 5/20 0.55
PPARG P37231 5/20 0.54
PPARA Q07869 3/20 0.54
TP53 P04637 1/20 0.46
RXFP1 Q9HBX9 1/20 0.46
NPC1 O15118 4/20 0.44
RAB9A P51151 4/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
SIRT2 Q8IXJ6 1/20 0.44
SIRT1 Q96EB6 1/20 0.44
SIRT3 Q9NTG7 1/20 0.44
TDP1 Q9NUW8 1/20 0.43
POLB P06746 1/20 0.43
CASP3 P42574 1/20 0.43
SENP8 Q96LD8 1/20 0.43
SENP7 Q9BQF6 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20839936 0.93 NR1H4 (0.65) NR1H4HSPH1F10PPARDPPARG
SCHEMBL20840618 0.91 NR1H4 (0.59) NR1H4HSPH1F10PPARDPPARG
SCHEMBL20839717 0.90 NR1H4 (0.70) NR1H4F10PPARDPPARGPPARA
SCHEMBL20839667 0.87 HSPH1 (0.73) NR1H4HSPH1F10PPARDPPARG
SCHEMBL20839988 0.86 NR1H4 (0.67) NR1H4F10PPARDPPARGPPARA
SCHEMBL20839675 0.84 NR1H4 (0.81) NR1H4PPARDPPARGPPARARXFP1
SCHEMBL20839731 0.83 NR1H4 (0.80) NR1H4HSPH1PPARDPPARGPPARA
SCHEMBL20839595 0.82 NR1H4 (0.66) NR1H4HSPH1PPARDPPARGPPARA
SCHEMBL20839781 0.80 NR1H4 (0.71) NR1H4HSPH1F10PPARDPPARG
SCHEMBL20839599 0.80 FADS1 (0.60) HSPH1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019057969-A1 DUAL AGONISTS OF FXR AND PPARδ AND THEIR USES Johann Wolfgang Goethe-Universität (DE) 2019-03-28 WO disclosed