SCHEMBL20839719

SCHEMBL20839719

O=C(O)CCc1cccc(NC(=O)c2ccccc2NC(=O)C2=Cc3cccc(Cl)c3OC2)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 10/20 0.54
PPARD Q03181 9/20 0.54
PPARG P37231 7/20 0.54
PPARA Q07869 7/20 0.54
HSPH1 Q92598 1/20 0.47
MAOA P21397 2/20 0.47
MAOB P27338 2/20 0.47
KDM4E B2RXH2 2/20 0.45
MEN1 O00255 2/20 0.45
ALDH1A1 P00352 2/20 0.45
MAPT P10636 2/20 0.45
HPGD P15428 2/20 0.45
KMT2A Q03164 2/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
SIRT1 Q96EB6 1/20 0.44
ABCG2 Q9UNQ0 1/20 0.43
CYP3A4 P08684 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20839984 0.90 NR1H4 (0.55) NR1H4PPARDPPARGPPARAHSPH1
SCHEMBL20839506 0.90 NR1H4 (0.57) NR1H4PPARDPPARGPPARAHSPH1
SCHEMBL20839603 0.88 HTT (0.44) NR1H4PPARDPPARGPPARAMAOA
SCHEMBL20839742 0.88 NR1H4 (0.57) NR1H4PPARDPPARGPPARAHSPH1
SCHEMBL20839660 0.87 NPC1 (0.56) NR1H4PPARDPPARGPPARAMAOB
SCHEMBL20839654 0.86 MEN1 (0.62) NR1H4PPARDPPARGPPARAHSPH1
SCHEMBL20839968 0.83 NR1H4 (0.56) NR1H4PPARDPPARGPPARAHSPH1
SCHEMBL20839662 0.83 NR1H4 (0.55) NR1H4PPARDPPARGPPARAHSPH1
SCHEMBL20839696 0.83 NR1H4 (0.55) NR1H4PPARDPPARGPPARAMAOA
SCHEMBL20839749 0.79 MAOB (0.59) NR1H4PPARDPPARGPPARAMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019057969-A1 DUAL AGONISTS OF FXR AND PPARδ AND THEIR USES Johann Wolfgang Goethe-Universität (DE) 2019-03-28 WO disclosed
WO-2019057969-A1 DUAL AGONISTS OF FXR AND PPARδ AND THEIR USES Johann Wolfgang Goethe-Universität (DE) 2019-03-28 WO disclosed