SCHEMBL20839742

SCHEMBL20839742

O=C(O)CCc1cccc(NC(=O)c2ccccc2NC(=O)C2=Cc3ccccc3OC2)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 9/20 0.57
PPARD Q03181 7/20 0.57
PPARG P37231 6/20 0.57
PPARA Q07869 6/20 0.57
MAOB P27338 4/20 0.57
MAOA P21397 3/20 0.57
NPC1 O15118 4/20 0.52
MAPT P10636 4/20 0.52
RAB9A P51151 4/20 0.52
SMN1; SMN2 Q16637 4/20 0.52
MEN1 O00255 3/20 0.52
KMT2A Q03164 3/20 0.52
KDM4E B2RXH2 3/20 0.52
ALDH1A1 P00352 2/20 0.52
HPGD P15428 2/20 0.52
HTT P42858 1/20 0.50
NFKB1 P19838 3/20 0.49
NFKB2 Q00653 3/20 0.49
RELA Q04206 3/20 0.49
CASP3 P42574 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20839968 0.91 NR1H4 (0.56) NR1H4PPARDPPARGPPARAMAOB
SCHEMBL20839749 0.91 MAOB (0.59) NR1H4PPARDPPARGPPARAMAOB
SCHEMBL20839696 0.90 NR1H4 (0.55) NR1H4PPARDPPARGPPARAMAOB
SCHEMBL20839662 0.90 NR1H4 (0.55) NR1H4PPARDPPARGPPARAMAOB
SCHEMBL20839654 0.90 MEN1 (0.62) NR1H4PPARDPPARGPPARAMAOB
SCHEMBL20839984 0.89 NR1H4 (0.55) NR1H4PPARDPPARGPPARAMAOB
SCHEMBL20839506 0.88 NR1H4 (0.57) NR1H4PPARDPPARGPPARAMAOB
SCHEMBL20839719 0.88 NR1H4 (0.54) NR1H4PPARDPPARGPPARAMAOB
SCHEMBL20839499 0.88 HTT (0.56) NR1H4PPARDPPARGPPARAMAOB
SCHEMBL20839983 0.88 NR1H4 (0.56) NR1H4PPARDPPARGPPARAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019057969-A1 DUAL AGONISTS OF FXR AND PPARδ AND THEIR USES Johann Wolfgang Goethe-Universität (DE) 2019-03-28 WO disclosed
WO-2019057969-A1 DUAL AGONISTS OF FXR AND PPARδ AND THEIR USES Johann Wolfgang Goethe-Universität (DE) 2019-03-28 WO disclosed